Steroid regulation: An overlooked aspect of tolerance and chronic rejection in kidney transplantation

Mol Cell Endocrinol. 2018 Sep 15:473:205-216. doi: 10.1016/j.mce.2018.01.021. Epub 2018 Feb 7.

Abstract

Steroid conversion (HSD11B1, HSD11B2, H6PD) and receptor genes (NR3C1, NR3C2) were examined in kidney-transplant recipients with "operational tolerance" and chronic rejection (CR), independently and within the context of 88 tolerance-associated genes. Associations with cellular types were explored. Peripheral whole-blood gene-expression levels (RT-qPCR-based) and cell counts were adjusted for immunosuppressant drug intake. Tolerant (n = 17), stable (n = 190) and CR patients (n = 37) were compared. Healthy controls (n = 14) were used as reference. The anti-inflammatory glucocorticoid receptor (NR3C1) and the cortisol-activating HSD11B1 and H6PD genes were up-regulated in CR and were lowest in tolerant patients. The pro-inflammatory mineralocorticoid gene (NR3C2) was downregulated in stable and CR patients. NR3C1 was associated with neutrophils and NR3C2 with T-cells. Steroid conversion and receptor genes, alone, enabled classification of tolerant patients and were major contributors to gene-expression signatures of both, tolerance and CR, alongside known tolerance-associated genes, revealing a key role of steroid regulation and response in kidney transplantation.

Keywords: Chronic rejection; Kidney; Steroid conversion; Steroid receptor genes; Tolerance; Transplantation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Area Under Curve
  • Cell Count
  • Chronic Disease
  • Gene Expression Regulation / drug effects
  • Graft Rejection / etiology*
  • Graft Rejection / genetics
  • Graft Rejection / immunology*
  • Humans
  • Immune Tolerance* / drug effects
  • Immune Tolerance* / genetics
  • Kidney Transplantation / adverse effects*
  • Multivariate Analysis
  • Prednisolone / administration & dosage
  • Prednisolone / pharmacology
  • Probability
  • Protein Isoforms / metabolism
  • Receptors, Glucocorticoid / metabolism
  • Regression Analysis
  • Steroids / pharmacology*
  • Up-Regulation / drug effects

Substances

  • Protein Isoforms
  • Receptors, Glucocorticoid
  • Steroids
  • Prednisolone