Pharmacological Inhibition of Necroptosis Protects from Dopaminergic Neuronal Cell Death in Parkinson's Disease Models

Cell Rep. 2018 Feb 20;22(8):2066-2079. doi: 10.1016/j.celrep.2018.01.089.

Abstract

Dysfunctions in mitochondrial dynamics and metabolism are common pathological processes associated with Parkinson's disease (PD). It was recently shown that an inherited form of PD and dementia is caused by mutations in the OPA1 gene, which encodes for a key player in mitochondrial fusion and structure. iPSC-derived neural cells from these patients exhibited severe mitochondrial fragmentation, respiration impairment, ATP deficits, and heightened oxidative stress. Reconstitution of normal levels of OPA1 in PD-derived neural cells normalized mitochondria morphology and function. OPA1-mutated neuronal cultures showed reduced survival in vitro. Intriguingly, selective inhibition of necroptosis effectively rescued this survival deficit. Additionally, dampening necroptosis in MPTP-treated mice protected from DA neuronal cell loss. This human iPSC-based model captures both early pathological events in OPA1 mutant neural cells and the beneficial effects of blocking necroptosis, highlighting this cell death process as a potential therapeutic target for PD.

Keywords: OPA1; Parkinson’s disease; apoptosis; cell death; iPSCs; mitochondria; necroptosis; necrosis; neurodegeneration.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine
  • Animals
  • Apoptosis / drug effects*
  • Cell Differentiation / drug effects
  • Disease Models, Animal
  • Dopaminergic Neurons / drug effects
  • Dopaminergic Neurons / pathology*
  • GTP Phosphohydrolases / genetics
  • Induced Pluripotent Stem Cells / drug effects
  • Induced Pluripotent Stem Cells / metabolism
  • Lysosomes / drug effects
  • Lysosomes / metabolism
  • Male
  • Membrane Potential, Mitochondrial / drug effects
  • Mice, Inbred C57BL
  • Mitochondria / drug effects
  • Mitochondria / metabolism
  • Mutation / genetics
  • Necrosis
  • Neural Stem Cells / drug effects
  • Neural Stem Cells / metabolism
  • Neuroprotective Agents / pharmacology*
  • Oxidative Stress / drug effects
  • Parkinson Disease / pathology*
  • Small Molecule Libraries / pharmacology

Substances

  • Neuroprotective Agents
  • Small Molecule Libraries
  • 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine
  • GTP Phosphohydrolases
  • OPA1 protein, human