Peroxisome Proliferator-Activated Receptor γ and Its Role in Adipocyte Homeostasis and Thiazolidinedione-Mediated Insulin Sensitization

Mol Cell Biol. 2018 Apr 30;38(10):e00677-17. doi: 10.1128/MCB.00677-17. Print 2018 May 15.

Abstract

Adipose tissue is a dynamic organ that makes critical contributions to whole-body metabolic homeostasis. Although recent studies have revealed that different fat depots have distinct molecular signatures, metabolic functions and adipogenic mechanisms, peroxisome proliferator-activated receptor γ (PPARγ) is still widely viewed as the master regulator of adipogenesis and critical for maintaining mature adipocyte function. Using an inducible, adipocyte-specific knockout system, we explored the role of PPARγ in mature adipocytes in vivo Short-term PPARγ deficiency in adipocytes reduces whole-body insulin sensitivity, but adipocytes are viable both in vitro and in vivo However, after exposure to a high-fat diet, even short-term PPARγ deficiency leads to rapid adipocyte death. When mature adipocytes are depleted of both PPARγ and CCAAT-enhancer-binding protein α (C/EBPα), they are rapidly depleted of lipids and undergo adipocyte death, both in vitro and in vivo Surprisingly, although thiazolidinediones (TZDs; PPARγ agonists) are thought to act mainly on PPARγ, PPARγ in adipocytes is not required for the whole-body insulin-sensitizing effect of TZDs. This offers new mechanistic aspects of PPARγ/TZD action and its effect on whole-body metabolic homeostasis.

Keywords: C/EBPα; PPARγ; adipocyte; adipose tissue; inducible knockout; insulin sensitization; mouse model; obesity; thiazolidinedione.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adipocytes / metabolism*
  • Adipogenesis / physiology
  • Adipose Tissue / physiology
  • Animals
  • CCAAT-Enhancer-Binding Protein-alpha / metabolism
  • Homeostasis / physiology
  • Insulin / metabolism
  • Insulin Resistance / physiology*
  • Mice
  • Mice, Inbred C57BL
  • PPAR gamma / physiology*
  • Thiazolidinediones / pharmacology
  • Transcription Factors

Substances

  • CCAAT-Enhancer-Binding Protein-alpha
  • Insulin
  • PPAR gamma
  • Thiazolidinediones
  • Transcription Factors
  • 2,4-thiazolidinedione