Optimized Camellia sinensis var. sinensis, Ilex paraguariensis, and Aspalathus linearis blend presents high antioxidant and antiproliferative activities in a beverage model

Food Chem. 2018 Jul 15:254:348-358. doi: 10.1016/j.foodchem.2018.02.021. Epub 2018 Feb 6.

Abstract

A statistical optimization study was conducted to obtain a tea containing fermented rooibos (Aspalathus linearis), white tea (Camellia sinensis var. sinensis), and roasted mate (Ilex paraguariensis). An optimal combination of these species was proposed. This optimized tea inhibited 64% the lipoperoxidation in vitro and presented a high phenolic content, especially kaempferol, (+)-catechin, (-)-epicatechin, rutin, (-)-epigallocatechin, and (-)-epicatechin-2-O-gallate. Indeed, the antioxidant effect was confirmed by decreasing 30% the reactive oxygen species generation in human hepatoma carcinoma cells (HepG2, 100 and 240 µg/mL). In the cell viability assay, the GI50 for human colorectal adenocarcinoma epithelial cells (Caco-2) was about 547 µg/mL and 481 µg/mL for HepG2. The pasteurization process (65 °C/30 min) did not affect the total phenolic content and antioxidant activity of the optimized tea formulation. The sensory test indicated an acceptability index of 78%, showing that the analytical approach adopted was feasible to develop a phenolic-rich beverage.

Keywords: Antimicrobials; Cell viability; Desirability function; IC(50); Phenolic compounds; Reactive oxygen species; Response surface methodology.

MeSH terms

  • Adolescent
  • Adult
  • Anti-Infective Agents / pharmacology
  • Antioxidants / analysis
  • Antioxidants / pharmacology*
  • Aspalathus / chemistry*
  • Beverages
  • Caco-2 Cells
  • Camellia sinensis / chemistry*
  • Female
  • Hep G2 Cells
  • Humans
  • Ilex paraguariensis / chemistry*
  • Male
  • Middle Aged
  • Pasteurization
  • Phenols / analysis
  • Plant Extracts / pharmacology
  • Reactive Oxygen Species / metabolism
  • Taste
  • Teas, Herbal* / analysis

Substances

  • Anti-Infective Agents
  • Antioxidants
  • Phenols
  • Plant Extracts
  • Reactive Oxygen Species
  • Teas, Herbal