Decreased cAMP Level and Decreased Downregulation of β1-Adrenoceptor Expression in Therapeutic Hypothermia-Resuscitated Myocardium Are Associated With Improved Post-Resuscitation Myocardial Function

J Am Heart Assoc. 2018 Mar 23;7(6):e006573. doi: 10.1161/JAHA.117.006573.

Abstract

Background: Epinephrine administered during cardiopulmonary resuscitation (CPR) is associated with severe post-resuscitation myocardial dysfunction. We previously demonstrated that therapeutic hypothermia reduced the severity of post-resuscitation myocardial dysfunction caused by epinephrine; however, the relationship between myocardial adrenoceptor expression and myocardial protective effects by hypothermia remains unclear.

Methods and results: Rats weighing between 450 and 550 g were randomized into 5 groups: (1) normothermic placebo, (2) normothermic epinephrine, (3) hypothermic placebo, (4) hypothermic epinephrine, and (5) sham (not subject to cardiac arrest and resuscitation). Ventricular fibrillation was induced and untreated for 8 minutes for all other groups. Hypothermia was initiated coincident with the start of CPR and maintained at 33±0.2°C for 4 hours. Placebo or epinephrine was administered 5 minutes after the start of CPR and 3 minutes before defibrillation. Post-resuscitation ejection fraction was measured hourly for 4 hours then hearts were harvested. Epinephrine increased coronary perfusion pressure during CPR (27±6 mm Hg versus 21±2 mm Hg P<0.05). Post-resuscitation myocardial function was impaired in the normothermic epinephrine group compared with other groups. The concentration of myocardial cAMP doubled in the normothermic epinephrine group (655.06±447.63 μmol/L) compared with the hypothermic epinephrine group (302.51±97.98 μmol/L; P<0.05). Myocardial β1-adrenoceptor expression decreased with normothermia cardiac arrest but not with hypothermia regardless of epinephrine.

Conclusions: Epinephrine, administered during normothermic CPR, increased the severity of post-resuscitation myocardial dysfunction. This adverse effect was inhibited by intra-arrest hypothermia resuscitation. Declined cAMP with more preserved β1-adrenoceptors in hypothermia-resuscitated myocardium is associated with improved post-resuscitated myocardial function in vivo.

Keywords: CPR; adrenoceptor; epinephrine; hypothermia; post‐resuscitation.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenergic Agonists / administration & dosage
  • Adrenergic Agonists / toxicity*
  • Animals
  • Cardiopulmonary Resuscitation / adverse effects*
  • Cardiopulmonary Resuscitation / methods
  • Cyclic AMP / metabolism*
  • Disease Models, Animal
  • Epinephrine / administration & dosage
  • Epinephrine / toxicity*
  • Heart Arrest / metabolism
  • Heart Arrest / physiopathology
  • Heart Arrest / therapy*
  • Hypothermia, Induced*
  • Male
  • Myocardium / metabolism*
  • Rats, Sprague-Dawley
  • Receptors, Adrenergic, beta-1 / metabolism*
  • Recovery of Function
  • Time Factors
  • Ventricular Function / drug effects*

Substances

  • Adrb1 protein, rat
  • Adrenergic Agonists
  • Receptors, Adrenergic, beta-1
  • Cyclic AMP
  • Epinephrine