Generation and testing of clinical-grade exosomes for pancreatic cancer

JCI Insight. 2018 Apr 19;3(8):e99263. doi: 10.1172/jci.insight.99263.

Abstract

Exosomes are extracellular vesicles produced by all cells with a remarkable ability to efficiently transfer genetic material, including exogenously loaded siRNA, to cancer cells. Here, we report on a bioreactor-based, large-scale production of clinical-grade exosomes employing good manufacturing practice (GMP) standards. A standard operating procedure was established to generate engineered exosomes with the ability to target oncogenic Kras (iExosomes). The clinical-grade GMP iExosomes were tested in multiple in vitro and in vivo studies to confirm suppression of oncogenic Kras and an increase in the survival of several mouse models with pancreatic cancer. We perform studies to determine the shelf life, biodistribution, toxicology profile, and efficacy in combination with chemotherapy to inform future clinical testing of GMP iExosomes. Collectively, this report illustrates the process and feasibility of generating clinical-grade exosomes for various therapies of human diseases.

Keywords: Cancer gene therapy; Oncology.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line, Tumor / drug effects
  • Cell Line, Tumor / metabolism*
  • Disease Models, Animal
  • Drug Therapy / methods
  • Drug Therapy, Combination / methods
  • Exosomes / genetics*
  • Female
  • Genetic Therapy / methods
  • Male
  • Mice
  • Mice, Inbred C57BL / genetics
  • Pancreatic Neoplasms / drug therapy
  • Pancreatic Neoplasms / genetics*
  • Pancreatic Neoplasms / metabolism
  • Pancreatic Neoplasms / veterinary
  • Proto-Oncogene Proteins p21(ras) / genetics*
  • RNA, Small Interfering / genetics*

Substances

  • RNA, Small Interfering
  • Proto-Oncogene Proteins p21(ras)