Abstract
R2TP is an HSP90 co-chaperone that assembles important macro-molecular machineries. It is composed of an RPAP3-PIH1D1 heterodimer, which binds the two essential AAA+ATPases RUVBL1/RUVBL2. Here, we resolve the structure of the conserved C-terminal domain of RPAP3, and we show that it directly binds RUVBL1/RUVBL2 hexamers. The human genome encodes two other proteins bearing RPAP3-C-terminal-like domains and three containing PIH-like domains. Systematic interaction analyses show that one RPAP3-like protein, SPAG1, binds PIH1D2 and RUVBL1/2 to form an R2TP-like complex termed R2SP. This co-chaperone is enriched in testis and among 68 of the potential clients identified, some are expressed in testis and others are ubiquitous. One substrate is liprin-α2, which organizes large signaling complexes. Remarkably, R2SP is required for liprin-α2 expression and for the assembly of liprin-α2 complexes, indicating that R2SP functions in quaternary protein folding. Effects are stronger at 32 °C, suggesting that R2SP could help compensating the lower temperate of testis.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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ATPases Associated with Diverse Cellular Activities / metabolism*
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Adaptor Proteins, Signal Transducing / metabolism
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Antigens, Surface / metabolism
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Apoptosis Regulatory Proteins / genetics
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Apoptosis Regulatory Proteins / metabolism*
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Carrier Proteins / genetics
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Carrier Proteins / metabolism*
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Cell Line
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DNA Helicases / metabolism*
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GTP-Binding Proteins / metabolism
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HEK293 Cells
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HSP90 Heat-Shock Proteins / metabolism*
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HeLa Cells
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Humans
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Male
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Membrane Proteins / metabolism
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Molecular Chaperones / metabolism*
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Protein Binding
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Protein Folding
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Protein Structure, Secondary
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Signal Transduction
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Testis / metabolism*
Substances
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Adaptor Proteins, Signal Transducing
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Antigens, Surface
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Apoptosis Regulatory Proteins
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Carrier Proteins
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HSP90 Heat-Shock Proteins
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Membrane Proteins
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Molecular Chaperones
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PIH1D1 protein, human
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PPFIA2 protein, human
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RPAP3 protein, human
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GTP-Binding Proteins
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SPAG1 protein, human
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ATPases Associated with Diverse Cellular Activities
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DNA Helicases
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RUVBL1 protein, human
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RUVBL2 protein, human