Blocking Properdin Prevents Complement-Mediated Hemolytic Uremic Syndrome and Systemic Thrombophilia

J Am Soc Nephrol. 2018 Jul;29(7):1928-1937. doi: 10.1681/ASN.2017121244. Epub 2018 Jun 1.

Abstract

Background Properdin (P) is a positive regulator of the alternative pathway of complement activation. Although P inhibition is expected and has been shown to ameliorate the alternative pathway of complement-mediated tissue injury in several disease models, it unexpectedly exacerbated renal injury in a murine model of C3 glomerulopathy. The role of P in atypical hemolytic uremic syndrome (aHUS) is uncertain.Methods We blocked P function by genetic deletion or mAb-mediated inhibition in mice carrying a factor H (FH) point mutation, W1206R (FHR/R), that causes aHUS and systemic thrombophilia with high mortality.Results P deficiency completely rescued FHR/R mice from premature death and prevented thrombocytopenia, hemolytic anemia, and renal disease. It also eliminated macrovessel thrombi that were prevalent in FHR/R mice. All mice that received a function-blocking anti-P mAb for 8 weeks survived the experimental period and appeared grossly healthy. Platelet counts and hemoglobin levels were significantly improved in FHR/R mice after 4 weeks of anti-P mAb treatment. One half of the FHR/R mice treated with an isotype control mAb but none of the anti-P mAb-treated mice developed stroke-related neurologic disease. Anti-P mAb-treated FHR/R mice showed largely normal renal histology, and residual liver thrombi were detected in only three of 15 treated mice.Conclusions These results contrast with the detrimental effect of P inhibition observed in a murine model of C3 glomerulopathy and suggest that P contributes critically to aHUS pathogenesis. Inhibition of P in aHUS may be of therapeutic benefit.

Keywords: Immunology and pathology; complement; hemolytic uremic syndrome.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibodies, Monoclonal / therapeutic use
  • Atypical Hemolytic Uremic Syndrome / drug therapy
  • Atypical Hemolytic Uremic Syndrome / genetics*
  • Atypical Hemolytic Uremic Syndrome / prevention & control
  • Complement C3 / metabolism*
  • Complement C9 / metabolism*
  • Complement Factor H / genetics
  • Complement Pathway, Alternative
  • Female
  • Fibrin / metabolism
  • Hemoglobins / metabolism
  • Kidney / metabolism
  • Kidney / pathology
  • Male
  • Mice
  • Mice, Knockout
  • Platelet Count
  • Properdin / deficiency
  • Properdin / genetics*
  • Properdin / immunology
  • Thrombophilia / genetics*
  • Thrombophilia / prevention & control
  • Thrombosis / prevention & control

Substances

  • Antibodies, Monoclonal
  • Complement C3
  • Complement C9
  • Hemoglobins
  • Properdin
  • Complement Factor H
  • Fibrin