In vitro thrombolytic activity of a purified fibrinolytic enzyme from Chlorella vulgaris

J Chromatogr B Analyt Technol Biomed Life Sci. 2018 Aug 15:1092:524-529. doi: 10.1016/j.jchromb.2018.04.040. Epub 2018 Apr 24.

Abstract

A fibrinolytic enzyme was produced by microalga Chlorella vulgaris cultivated in autotrophic and mixotrophic conditions added corn steep liquor, purified by a single chromatographic step, then biochemical characterization and in vitro thrombolytic activity was performed. Maximum cell concentration (1637.45 ± 15 mg L-1) and productivity (181.93 mg L-1 day-1) was obtained in mixotrophic culture using 1% corn steep liquor. Enzyme-extracted microalgal biomass was purified by acetone precipitation and DEAE Sephadex anion exchange chromatography up to 2 fold with recovery of 4.0%. After purification, fibrinolytic activity was 1834.6 U mg-1 and 226.86 mm2 by spectrophotometry and fibrin plate assays, respectively. SDS-PAGE results exhibited a protein band of about 45 kDa and fibrinolytic band was detected by fibrin zymography. Enzyme activity was enhanced in the presence of Fe2+ and inhibited by phenylmethane sulfonyl fluoride (PMSF) and ethylenediamine tetracetic acid (EDTA), which suggest it to be a metal-dependent serine protease. The extract also showed a red blood cell lysis <4% and in vitro thrombolytic activity of 25.6% in 90 min of reaction. These results indicate that the fibrinolytic enzyme from C. vulgaris may have potential applications in the prevention and treatment of thrombosis.

Keywords: Chlorella vulgaris; Chromatography; Corn Steep Liquor; Fibrinolytic enzyme; Thrombolytic activity.

MeSH terms

  • Chlorella vulgaris / enzymology*
  • Chromatography, Ion Exchange / methods
  • Erythrocytes / drug effects
  • Fibrin / metabolism*
  • Fibrinolytic Agents* / chemistry
  • Fibrinolytic Agents* / isolation & purification
  • Fibrinolytic Agents* / pharmacology
  • Hemolysis / drug effects
  • Humans
  • Plant Proteins* / chemistry
  • Plant Proteins* / isolation & purification
  • Plant Proteins* / pharmacology

Substances

  • Fibrinolytic Agents
  • Plant Proteins
  • Fibrin