Emergence of Integrase Resistance Mutations During Initial Therapy Containing Dolutegravir

Clin Infect Dis. 2018 Aug 16;67(5):791-794. doi: 10.1093/cid/ciy228.

Abstract

Dolutegravir (DTG) is a preferred drug for initial treatment of human immunodeficiency virus type 1 infection. We present next-generation sequencing analysis of integrase genotypes during a period of virologic failure in a treatment-naive man who initiated tenofovir disoproxil fumarate/emtricitabine plus DTG.

Publication types

  • Case Reports
  • Research Support, N.I.H., Extramural

MeSH terms

  • Antiretroviral Therapy, Highly Active
  • Drug Resistance, Viral*
  • Genotype
  • HIV Infections / drug therapy*
  • HIV Integrase Inhibitors / therapeutic use*
  • HIV-1 / drug effects*
  • HIV-1 / enzymology
  • HIV-1 / genetics
  • Heterocyclic Compounds, 3-Ring / therapeutic use*
  • Humans
  • Integrases / genetics*
  • Male
  • Middle Aged
  • Mutation
  • Oxazines
  • Piperazines
  • Pyridones
  • Sequence Analysis, DNA
  • Treatment Failure

Substances

  • HIV Integrase Inhibitors
  • Heterocyclic Compounds, 3-Ring
  • Oxazines
  • Piperazines
  • Pyridones
  • dolutegravir
  • Integrases