Ability of various alkylating agents to induce adaptive and SOS responses: a study with lacZ fusion

Mutat Res. 1985 Sep;146(2):149-54. doi: 10.1016/0167-8817(85)90005-7.

Abstract

We used alkA'-lacZ' and umuC'-lacZ' fused genes and determined the ability of various alkylating agents to induce adaptive and SOS responses. The degree of induction of expression of these genes was quantitatively measured by a simple colorimetric assay of beta-galactosidase activity. SN1 type methylating agents, such as N-methyl-N'-nitro-N-nitrosoguanidine and N-methyl-N-nitrosourea, were more effective inducers for the alkA than for the umuC system, while SN1 type ethylating agents, such as N-ethyl-N'-nitro-N-nitrosoguanidine and N-ethyl-N-nitrosourea, were more potent inducers for the umuC than for the alkA system. Similar but less striking effects on the two systems were obtained with SN2 type alkylating agents.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkylating Agents / pharmacology*
  • Bacterial Proteins / genetics
  • DNA Glycosylases*
  • DNA Ligases / biosynthesis*
  • DNA Ligases / genetics
  • DNA Repair*
  • Dose-Response Relationship, Drug
  • Enzyme Induction / drug effects
  • Escherichia coli / genetics
  • Escherichia coli / metabolism
  • Ethylnitrosourea / pharmacology
  • Genes, Bacterial
  • Genes, Synthetic / drug effects
  • Guanine / metabolism
  • Lac Operon*
  • Methylation
  • Methylnitronitrosoguanidine / pharmacology
  • Methylnitrosourea / pharmacology
  • N-Glycosyl Hydrolases / genetics
  • Polynucleotide Ligases / biosynthesis*
  • beta-Galactosidase / biosynthesis
  • beta-Galactosidase / genetics

Substances

  • Alkylating Agents
  • Bacterial Proteins
  • Methylnitronitrosoguanidine
  • Guanine
  • Methylnitrosourea
  • beta-Galactosidase
  • 3-methyladenine-DNA glycosylase
  • DNA Glycosylases
  • N-Glycosyl Hydrolases
  • DNA Ligases
  • Polynucleotide Ligases
  • Ethylnitrosourea