Protective effects of dopamine D2/D3 receptor agonist piribedil on learning and memory of rats exposed to global cerebral ischemia-reperfusion

Neurosci Lett. 2018 Sep 25:684:181-186. doi: 10.1016/j.neulet.2018.08.011. Epub 2018 Aug 11.

Abstract

Global cerebral ischemia-reperfusion (GCI/R) may occur after any of several clinical conditions such as cardiac arrest and anesthetic accident. Some dopamine receptor agonists possess neuroprotective effects. However, some of them may produce side effects during treatment. Piribedil, which is a dopamine D2/D3 receptor agonist, has fewer side effects and is well tolerated. This study investigated the effects of piribedil on learning and memory of rats with GCI/R according to modified neurological severity score (mNSS) scoring and Morris water maze test (MWM). Rats with GCI/R were treated with piribedil 25 or 50 mg/kg/d, and mNSS was performed at 6 h, 1 day, 3 days, and 1 and 2 weeks after injury. The MWM test was employed to evaluate learning and memory of rats at 1 and 2 weeks after injury. The results showed treatment with piribedil reduced the mNSS score and prolonged the time in the target quadrant compared with untreated rats although no obvious differences of the 25 and 50 mg/kg/d piribedil intervention groups were observed statistically. Piribedil is effective in improving the neurological function and learning and memory of rats after GCI/R.

Keywords: Behavior; Cerebral ischemia-reperfusion injury; Learning memory; Morris water maze; Piribedil.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Brain Ischemia / drug therapy*
  • Brain Ischemia / physiopathology
  • Dopamine Agonists / pharmacology
  • Dopamine Agonists / therapeutic use*
  • Dose-Response Relationship, Drug
  • Male
  • Maze Learning / drug effects*
  • Maze Learning / physiology
  • Memory / drug effects*
  • Memory / physiology
  • Neuroprotective Agents / pharmacology
  • Neuroprotective Agents / therapeutic use
  • Piribedil / pharmacology
  • Piribedil / therapeutic use*
  • Random Allocation
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Dopamine D2 / agonists*
  • Receptors, Dopamine D3 / agonists*
  • Reperfusion Injury / drug therapy
  • Reperfusion Injury / physiopathology
  • Treatment Outcome

Substances

  • Dopamine Agonists
  • Neuroprotective Agents
  • Receptors, Dopamine D2
  • Receptors, Dopamine D3
  • Piribedil