A new mechanism for LKB1 activation

Mol Cell Oncol. 2018 Apr 10;5(3):e1035691. doi: 10.1080/23723556.2015.1035691. eCollection 2018.

Abstract

Liver kinase B1 (LKB1, also known as serine/threonine kinase 11, STK11) has been thought to be a constitutively active tumor suppressor that is activated by forming an active complex. Very recently, a new post-translational modification on LKB1 was identified that can regulate LKB1 activation and LKB1-mediated cancer cell survival under energy stress.

Keywords: AMPK; LKB1; mechanisms of oncogenesis and tumor progression; ras; skp2; ubiquitination.

Grants and funding

This study was supported by CPRIT grant, NIH RO1 grants, R. Lee Clark Award, and MD Anderson prostate moonshot program to H.-K.L.