Antibody drug conjugates in thoracic malignancies

Lung Cancer. 2018 Oct:124:260-269. doi: 10.1016/j.lungcan.2018.07.001. Epub 2018 Jul 19.

Abstract

Antibody drug conjugates (ADCs) have the potential to alter the efficacy: toxicity ratio of cytotoxic therapy utilizing surface markers on cancer cells as antibody targets to preferentially deliver toxic payloads to tumor cells while limiting systemic toxicity. Multiple ADCs, differing in their antibody targets, cytotoxic payloads and linker molecules are currently being evaluated in non-small-cell lung cancer, small-cell lung cancer and malignant pleural mesothelioma. Here we review the available data in thoracic malignancies and the potential issues influencing the efficacy and toxicity of these approaches.

Keywords: Antibody drug conjugate; Mesothelioma; Non-small-cell lung cancer; Small-cell lung cancer; Thoracic malignancies.

Publication types

  • Research Support, N.I.H., Extramural
  • Review

MeSH terms

  • Carcinoma, Non-Small-Cell Lung / drug therapy*
  • Cytotoxicity, Immunologic
  • Humans
  • Immunoconjugates / therapeutic use*
  • Immunotherapy / methods*
  • Lung Neoplasms / drug therapy*
  • Mesothelioma / drug therapy*
  • Mesothelioma, Malignant
  • Pleural Neoplasms / drug therapy*
  • Thoracic Neoplasms / drug therapy*
  • Treatment Outcome

Substances

  • Immunoconjugates