Goniothalamin-Related Styryl Lactones: Isolation, Synthesis, Biological Activity and Mode of Action

Curr Med Chem. 2019;26(41):7372-7451. doi: 10.2174/0929867325666181009161439.

Abstract

This review covers the chemistry and biological aspects of goniothalamin-related styryl lactones isolated from natural sources. This family of secondary metabolites has been reported to display diverse uses in folk medicine, but only a limited number of these compounds have been throughly investigated regarding their biological profile. Herein, we cover the goniothalamin-related styryl lactones having a C6-C3-C4 framework which appeared in the literature for the first time in the period 2000-2017, and the reports on the synthesis, biological activity and mechanism of action which were published from 2007-2017.

Keywords: Goniothalamin; biological activity; isolation; mode of action; styryl lactones; synthesis..

Publication types

  • Review

MeSH terms

  • Drug Evaluation, Preclinical
  • Humans
  • Lactones / chemistry*
  • Pyrones / chemical synthesis
  • Pyrones / chemistry
  • Pyrones / pharmacology*
  • Structure-Activity Relationship

Substances

  • Lactones
  • Pyrones
  • goniothalamin