Meropenem-vaborbactam for adults with complicated urinary tract and other invasive infections

Expert Rev Anti Infect Ther. 2018 Dec;16(12):865-876. doi: 10.1080/14787210.2018.1542300. Epub 2018 Nov 5.

Abstract

Complicated urinary tract infections are increasingly caused by multidrug-resistant organisms. Carbapenem-resistant Enterobacteriaceae (CRE) constitute a rising threat among uropathogens with significant morbidity and mortality. Meropenem-vaborbactam is a novel carbapenem and cyclic boronic acid-based beta-lactamase inhibitor combination with potent activity against subtypes of CRE. Areas covered: This article reviews mechanisms of carbapenem resistance, existing treatment options for CRE, and the current evidence to support the use of meropenem-vaborbactam for the treatment of infections caused by subtypes of CRE including complicated urinary tract infections. Expert commentary: Meropenem-vaborbactam is a superior treatment option for infections secondary to Klebsiella pneumoniae carbapenemase (KPC)-producing CRE. It is associated with higher rates of treatment success and lower rates of toxicity than traditional agents and demonstrates a potentially higher barrier to acquired antimicrobial resistance than ceftazidime-avibactam. At present, meropenem-vaborbactam should be regarded as a preferred treatment option for invasive infections secondary to KPC-producing CRE.

Keywords: CRE; Complicated urinary tract infection; KPC; meropenem–vaborbactam; multidrug-resistant gram-negative organisms.

Publication types

  • Review

MeSH terms

  • Adult
  • Animals
  • Anti-Bacterial Agents / administration & dosage*
  • Anti-Bacterial Agents / adverse effects
  • Anti-Bacterial Agents / pharmacology
  • Boronic Acids / administration & dosage*
  • Boronic Acids / adverse effects
  • Boronic Acids / pharmacology
  • Carbapenem-Resistant Enterobacteriaceae / drug effects
  • Drug Combinations
  • Drug Resistance, Multiple, Bacterial
  • Enterobacteriaceae Infections / drug therapy
  • Enterobacteriaceae Infections / microbiology
  • Humans
  • Klebsiella pneumoniae / isolation & purification
  • Meropenem / administration & dosage*
  • Meropenem / adverse effects
  • Meropenem / pharmacology
  • Urinary Tract Infections / drug therapy
  • Urinary Tract Infections / microbiology

Substances

  • Anti-Bacterial Agents
  • Boronic Acids
  • Drug Combinations
  • vaborbactam
  • Meropenem