Patient-Specific iPSC-Derived Endothelial Cells Provide Long-Term Phenotypic Correction of Hemophilia A

Stem Cell Reports. 2018 Dec 11;11(6):1391-1406. doi: 10.1016/j.stemcr.2018.10.012. Epub 2018 Nov 8.

Abstract

We generated patient-specific disease-free induced pluripotent stem cells (iPSCs) from peripheral blood CD34+ cells and differentiated them into functional endothelial cells (ECs) secreting factor VIII (FVIII) for gene and cell therapy approaches to cure hemophilia A (HA), an X-linked bleeding disorder caused by F8 mutations. iPSCs were transduced with a lentiviral vector carrying FVIII transgene driven by an endothelial-specific promoter (VEC) and differentiated into bona fide ECs using an optimized protocol. FVIII-expressing ECs were intraportally transplanted in monocrotaline-conditioned non-obese diabetic (NOD) severe combined immune-deficient (scid)-IL2rγ null HA mice generating a chimeric liver with functional human ECs. Transplanted cells engrafted and proliferated in the liver along sinusoids, in the long term showed stable therapeutic FVIII activity (6%). These results demonstrate that the hemophilic phenotype can be rescued by transplantation of ECs derived from HA FVIII-corrected iPSCs, confirming the feasibility of cell-reprogramming strategy in patient-derived cells as an approach for HA gene and cell therapy.

Keywords: FVIII; cell and gene therapy; chimeric vasculature; endothelial cells; hemophilia A; induced pluripotent stem cells (iPSCs); lentiviral vectors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antigens, CD34 / metabolism
  • Biomarkers / metabolism
  • Cell Differentiation
  • Cell Proliferation
  • Disease Models, Animal
  • Endothelial Cells / cytology*
  • Endothelial Cells / transplantation
  • Factor VIII / metabolism
  • Fetal Blood / cytology
  • Fibroblasts / cytology
  • Hemophilia A / pathology
  • Hemophilia A / therapy*
  • Humans
  • Induced Pluripotent Stem Cells / cytology*
  • Induced Pluripotent Stem Cells / transplantation
  • Injections, Intraperitoneal
  • Liver / cytology
  • Mice
  • Microspheres
  • Phenotype
  • Portal Vein / metabolism
  • Tissue Donors

Substances

  • Antigens, CD34
  • Biomarkers
  • Factor VIII