Update on prevalence and mechanisms of resistance to linezolid, tigecycline and daptomycin in enterococci in Europe: Towards a common nomenclature

Drug Resist Updat. 2018 Sep:40:25-39. doi: 10.1016/j.drup.2018.10.002. Epub 2018 Nov 2.

Abstract

Vancomycin-resistant enterococci (VRE) are important nosocomial pathogens. Invasive VRE infections are difficult to treat since common therapeutic options including ampicillin and glycopeptides often fail. In vitro, most VRE remain susceptible to last-resort antibiotics such as linezolid, tigecycline and daptomycin. However, neither tigecycline nor linezolid act in a bactericidal manner, and daptomycin has proven activity only at high dosages licensed for treating enterococcal endocarditis. Despite these pharmacological and therapeutic limitations, reports on resistance to these last-resort drugs in VRE, and enterococci in general, have increased in recent years. In this review, we briefly recapitulate the current knowledge on the mode of action as well as the known and novel mechanisms of resistance and describe surveillance data on resistance to linezolid, tigecycline and daptomycin in enterococci. In addition, we also suggest a common nomenclature for designating enterococci and VRE with resistances to these important last-resort antibiotics.

Keywords: Daptomycin; Linezolid; Tigecycline; VRE; vanA; vanB.

Publication types

  • Review

MeSH terms

  • Anti-Bacterial Agents / pharmacology*
  • Anti-Bacterial Agents / therapeutic use
  • Bacterial Proteins / genetics
  • Carbon-Oxygen Ligases / genetics
  • Daptomycin / pharmacology*
  • Daptomycin / therapeutic use
  • Genotype
  • Gram-Positive Bacterial Infections / drug therapy
  • Humans
  • Linezolid / pharmacology*
  • Linezolid / therapeutic use
  • Microbial Sensitivity Tests
  • Mutation
  • Tigecycline / pharmacology*
  • Tigecycline / therapeutic use
  • Vancomycin Resistance / drug effects*
  • Vancomycin Resistance / genetics
  • Vancomycin-Resistant Enterococci / drug effects*
  • Vancomycin-Resistant Enterococci / genetics

Substances

  • Anti-Bacterial Agents
  • Bacterial Proteins
  • VanA ligase, Bacteria
  • Tigecycline
  • Carbon-Oxygen Ligases
  • Linezolid
  • Daptomycin