A new coumarin from Murraya alata activates TRPV1 channel

Nat Prod Res. 2020 Apr;34(8):1068-1073. doi: 10.1080/14786419.2018.1548455. Epub 2019 Jan 19.

Abstract

One new coumarin, muralatin R, was isolated from the leaves of Murraya alata Drake (Rutaceae). Its structure was elucidated by extensive analysis of the NMR and MS data, along with the specific rotation comparison. Muralatin R was found to be capable of activating the transient receptor potential vanilloid 1 (TRPV1) channel through desensitization mechanism. The results supply reference for clarification of the therapeutic basis and mechanism of action of Murraya plants for treating psychogenic pain or somatoform pain disorders.

Keywords: Murraya; Murraya alata; TRPV1 channel; coumarin; pain.

MeSH terms

  • Coumarins / chemistry
  • Coumarins / isolation & purification
  • Coumarins / pharmacology*
  • Humans
  • Magnetic Resonance Spectroscopy
  • Molecular Structure
  • Murraya / chemistry*
  • Pain / drug therapy
  • Plant Leaves / chemistry
  • Rutaceae
  • TRPV Cation Channels / drug effects*
  • TRPV Cation Channels / metabolism

Substances

  • Coumarins
  • TRPV Cation Channels
  • TRPV1 protein, human
  • coumarin