A defect of platelet release reaction in a patient with SLE: impaired platelet aggregation induced by phorbol ester with a normal phosphorylation of 40K protein

Scand J Haematol. 1986 Jan;36(1):44-54. doi: 10.1111/j.1600-0609.1986.tb02648.x.

Abstract

A 37-year-old female who suffered from SLE had a bleeding disorder. At the time of initial evaluation, the main disease demonstrated was a delta-storage pool deficiency. After this improved, a marked decrease of aggregation still remained, when induced by either ADP, epinephrine, collagen, A23187, thrombin, or PAF-acether. Although arachidonate-induced aggregation was slightly decreased, thromboxane B2 was produced normally in response to exogenous arachidonate. The patient's endoperoxides and/or thromboxane A2 aggregated aspirin-treated platelets, though her platelets were themselves unresponsive. Impaired aggregability induced by TPA (12-0-tetradecanoylphorbol-13-acetate) or OAG (1-oleoyl-2-acetyl-glycerol) was also found. However, the phosphorylation of P43 and P20 induced by several stimulators including CA++ ionophore was normal, using 32P-labelled platelets. It is suggested that TPA or OAG-induced platelet aggregation requires not only the phosphorylation of those proteins, but also another unknown mechanism after the phosphorylation, and that the platelet dysfunction of this patient was due to a defect of some mechanism involving Ca++ uptake or mobilization of cytoplasmic Ca++ from intracellular storage sites.

Publication types

  • Case Reports

MeSH terms

  • Adenosine Diphosphate / pharmacology
  • Adult
  • Arachidonic Acid
  • Arachidonic Acids / pharmacology
  • Blood Platelets / metabolism
  • Blood Platelets / ultrastructure
  • Blood Proteins / metabolism*
  • Calcimycin / pharmacology
  • Collagen / pharmacology
  • Diglycerides / pharmacology
  • Epinephrine / pharmacology
  • Female
  • Humans
  • Lupus Erythematosus, Systemic / blood*
  • Phorbols / pharmacology*
  • Phosphorylation
  • Platelet Activating Factor / pharmacology
  • Platelet Aggregation / drug effects*
  • Tetradecanoylphorbol Acetate / pharmacology*
  • Thrombin / pharmacology

Substances

  • Arachidonic Acids
  • Blood Proteins
  • Diglycerides
  • Phorbols
  • Platelet Activating Factor
  • Arachidonic Acid
  • Calcimycin
  • Adenosine Diphosphate
  • 1-oleoyl-2-acetylglycerol
  • Collagen
  • Thrombin
  • Tetradecanoylphorbol Acetate
  • Epinephrine