Removal of a Conserved Disulfide Bond Does Not Compromise Mechanical Stability of a VHH Antibody Complex

Nano Lett. 2019 Aug 14;19(8):5524-5529. doi: 10.1021/acs.nanolett.9b02062. Epub 2019 Jul 5.

Abstract

Single-domain VHH antibodies are promising reagents for medical therapy. A conserved disulfide bond within the VHH framework region is known to be critical for thermal stability, however, no prior studies have investigated its influence on the stability of VHH antibody-antigen complexes under mechanical load. Here, we used single-molecule force spectroscopy to test the influence of a VHH domain's conserved disulfide bond on the mechanical strength of the interaction with its antigen mCherry. We found that although removal of the disulfide bond through cysteine-to-alanine mutagenesis significantly lowered VHH domain denaturation temperature, it had no significant impact on the mechanical strength of the VHH:mCherry interaction with complex rupture occurring at ∼60 pN at 103-104 pN/sec regardless of disulfide bond state. These results demonstrate that mechanostable binding interactions can be built on molecular scaffolds that may be thermodynamically compromised at equilibrium.

Keywords: Antibodies; biophysics; disulfide bond; nanobody; single-molecule force spectroscopy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alanine / chemistry
  • Cysteine / chemistry*
  • Disulfides / chemistry*
  • Luminescent Proteins / chemistry
  • Models, Molecular
  • Protein Denaturation
  • Protein Domains
  • Protein Stability
  • Red Fluorescent Protein
  • Single-Domain Antibodies / chemistry*
  • Temperature
  • Thermodynamics

Substances

  • Disulfides
  • Luminescent Proteins
  • Single-Domain Antibodies
  • Cysteine
  • Alanine