SPRTN protease and checkpoint kinase 1 cross-activation loop safeguards DNA replication

Nat Commun. 2019 Jul 17;10(1):3142. doi: 10.1038/s41467-019-11095-y.

Abstract

The SPRTN metalloprotease is essential for DNA-protein crosslink (DPC) repair and DNA replication in vertebrate cells. Cells deficient in SPRTN protease exhibit DPC-induced replication stress and genome instability, manifesting as premature ageing and liver cancer. Here, we provide a body of evidence suggesting that SPRTN activates the ATR-CHK1 phosphorylation signalling cascade during physiological DNA replication by proteolysis-dependent eviction of CHK1 from replicative chromatin. During this process, SPRTN proteolyses the C-terminal/inhibitory part of CHK1, liberating N-terminal CHK1 kinase active fragments. Simultaneously, CHK1 full length and its N-terminal fragments phosphorylate SPRTN at the C-terminal regulatory domain, which stimulates SPRTN recruitment to chromatin to promote unperturbed DNA replication fork progression and DPC repair. Our data suggest that a SPRTN-CHK1 cross-activation loop plays a part in DNA replication and protection from DNA replication stress. Finally, our results with purified components of this pathway further support the proposed model of a SPRTN-CHK1 cross-activation loop.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Checkpoint Kinase 1 / metabolism
  • Checkpoint Kinase 1 / physiology*
  • DNA Breaks
  • DNA Replication
  • DNA-Binding Proteins / metabolism
  • DNA-Binding Proteins / physiology*
  • Genomic Instability
  • Models, Genetic*
  • Phosphorylation
  • Signal Transduction
  • Zebrafish / genetics
  • Zebrafish / metabolism

Substances

  • DNA-Binding Proteins
  • SPRTN protein, human
  • CHEK1 protein, human
  • Checkpoint Kinase 1