The Electronic Structure of the Metal Active Site Determines the Geometric Structure and Function of the Metalloregulator NikR

Biochemistry. 2019 Aug 27;58(34):3585-3591. doi: 10.1021/acs.biochem.9b00542. Epub 2019 Aug 14.

Abstract

NikR is a nickel-responsive metalloregulator protein that controls the level of Ni2+ ions in living cells. Previous studies have shown that NikR can bind a series of first-row transition metal ions but binds to DNA with high affinity only as a Ni2+ complex. To understand this metal selectivity, S K-edge X-ray absorption spectroscopy of NikR bound to different metal ions was used to evaluate the different electronic structures. The experimental results are coupled with density functional theory calculations on relevant models. This study shows that both the Zeff of the metal ion and the donor nature of the ligands determine the electronic structure of the metal site. This impacts the geometric structure of the metal site and thus the conformation of the protein. This contribution of electronic structure to geometric structure can be extended to other metal selective metalloregulators.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Catalytic Domain*
  • Escherichia coli / metabolism*
  • Escherichia coli Proteins / chemistry
  • Escherichia coli Proteins / metabolism*
  • Models, Molecular
  • Nickel
  • Protein Conformation
  • Repressor Proteins / chemistry
  • Repressor Proteins / metabolism*
  • X-Ray Absorption Spectroscopy

Substances

  • Escherichia coli Proteins
  • NikR protein, E coli
  • Repressor Proteins
  • Nickel