Safety assessment of the biotechnologically produced human-identical milk oligosaccharide 3-Fucosyllactose (3-FL)

Food Chem Toxicol. 2019 Dec:134:110818. doi: 10.1016/j.fct.2019.110818. Epub 2019 Sep 15.

Abstract

3-Fucosyllactose (3-FL), a highly abundant complex carbohydrate in human breast milk, functions as a prebiotic promoting early microbial colonization of the gut, increasing pathogen resistance and modulating immune responses. To investigate potential health benefits, 3-FL was produced by fermentation using a genetically modified E. coli K12 strain. The safety assessment of 3-FL included acute oral toxicity, in vitro and in vivo assessment of genetic toxicity, and a subchronic rodent feeding study. 3-FL was not acutely toxic at 5000 mg/kg bw, and there was no evidence of genetic toxicity in the bacterial reverse mutation test and chromosomal aberration assay. There was a repeatable statistically-significant trend in the 4-h S9-activated test conditions in the in vitro micronucleus assay; the confirmatory in vivo mouse micronucleus study was negative at all doses. Dietary subchronic exposure of rats to 3-FL (5% and 10%) did not produce any statistical or biologically-relevant differences in growth, food intake or efficiency, clinical observations, or clinical or anatomic pathology changes at average daily intakes of 5.98 and 7.27 g/kg bw/day for males and females, respectively. The weight of evidence from these studies support the safe use of 3-FL produced using biotechnology as a nutritional ingredient in foods.

Keywords: 3-FL; 3-Fucosyllactose; Human milk oligosaccharide; Infant formula; Nutritional ingredient; Safety.

MeSH terms

  • Animals
  • Biotechnology*
  • CHO Cells
  • Cricetulus
  • Dose-Response Relationship, Drug
  • Humans
  • Milk, Human / chemistry*
  • Mutagenicity Tests
  • No-Observed-Adverse-Effect Level
  • Oligosaccharides / chemical synthesis
  • Oligosaccharides / pharmacology*
  • Oligosaccharides / toxicity
  • Rats

Substances

  • Oligosaccharides
  • 3'-fucosyllactose