Pharmacokinetics of lisuride after subcutaneous infusion

J Neural Transm Suppl. 1988:27:71-4. doi: 10.1007/978-3-7091-8954-2_8.

Abstract

Six parkinsonian patients received a constant subcutaneous infusion of 60 micrograms lisuride per hour in the abdominal region for 2 hours. Plasma levels of the unchanged drug were measured by radio-immunoassay. During infusion, a steady state plasma level of 0.78 +/- 0.19 ng/ml was achieved. After discontinuation of the infusion, concentrations declined with a half-life of 1.4 +/- 0.4 hour. The total clearance of lisuride was 20 +/- 6 ml/min/kg. Due to the low interpatient variability of plasma levels, a good control of clinical effects is to be expected.

MeSH terms

  • Administration, Oral
  • Biological Availability
  • Ergolines / administration & dosage*
  • Humans
  • Infusion Pumps
  • Infusions, Parenteral
  • Injections, Intramuscular
  • Injections, Intravenous
  • Lisuride / administration & dosage*
  • Lisuride / blood
  • Lisuride / pharmacokinetics
  • Parkinson Disease / blood
  • Parkinson Disease / drug therapy
  • Time Factors

Substances

  • Ergolines
  • Lisuride