Thymosin β4 promotes autophagy and repair via HIF-1α stabilization in chronic granulomatous disease

Life Sci Alliance. 2019 Nov 12;2(6):e201900432. doi: 10.26508/lsa.201900432. Print 2019 Dec.

Abstract

Chronic granulomatous disease (CGD) is a genetic disorder of the NADPH oxidase characterized by increased susceptibility to infections and hyperinflammation associated with defective autophagy and increased inflammasome activation. Herein, we demonstrate that thymosin β4 (Tβ4), a g-actin sequestering peptide with multiple and diverse intracellular and extracellular activities affecting inflammation, wound healing, fibrosis, and tissue regeneration, promoted in human and murine cells noncanonical autophagy, a form of autophagy associated with phagocytosis and limited inflammation via the death-associated protein kinase 1. We further show that the hypoxia inducible factor-1 (HIF-1)α was underexpressed in CGD but normalized by Tβ4 to promote autophagy and up-regulate genes involved in mucosal barrier protection. Accordingly, inflammation and granuloma formation were impaired and survival increased in CGD mice with colitis or aspergillosis upon Tβ4 treatment or HIF-1α stabilization. Thus, the promotion of endogenous pathways of inflammation resolution through HIF-1α stabilization is druggable in CGD by Tβ4.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Actins / metabolism
  • Animals
  • Autophagy / physiology
  • DNA Repair
  • Female
  • Granulomatous Disease, Chronic / drug therapy*
  • Granulomatous Disease, Chronic / metabolism*
  • Granulomatous Disease, Chronic / pathology
  • Humans
  • Hypoxia-Inducible Factor 1, alpha Subunit / metabolism*
  • Male
  • Mice
  • Mice, Inbred C57BL
  • NADPH Oxidases / metabolism
  • RAW 264.7 Cells
  • Thymosin / pharmacology*

Substances

  • Actins
  • HIF1A protein, human
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • thymosin beta(4)
  • Thymosin
  • NADPH Oxidases