Targeting the Immune Complex-Bound Complement C3d Ligand as a Novel Therapy for Lupus

J Immunol. 2019 Dec 15;203(12):3136-3147. doi: 10.4049/jimmunol.1900620. Epub 2019 Nov 15.

Abstract

Humoral autoimmunity is central to the development of systemic lupus erythematosus (SLE). Complement receptor type 2 (CR2)/CD21 plays a key role in the development of high-affinity Abs and long-lasting memory to foreign Ags. When CR2 is bound by its primary C3 activation fragment-derived ligand, designated C3d, it coassociates with CD19 on B cells to amplify BCR signaling. C3d and CR2 also mediate immune complex binding to follicular dendritic cells. As the development of SLE involves subversion of normal B cell tolerance checkpoints, one might expect that CR2 ligation by C3d-bound immune complexes would promote development of SLE. However, prior studies in murine models of SLE using gene-targeted Cr2-/- mice, which lack both CR2 and complement receptor 1 (CR1), have demonstrated contradictory results. As a new approach, we developed a highly specific mouse anti-mouse C3d mAb that blocks its interaction with CR2. With this novel tool, we show that disruption of the critical C3d-CR2 ligand-receptor binding step alone substantially ameliorates autoimmunity and renal disease in the MRL/lpr model of SLE.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibodies, Monoclonal / immunology
  • Antibodies, Monoclonal / pharmacology
  • Antigen-Antibody Complex / immunology*
  • Antigen-Antibody Complex / metabolism
  • Autoantibodies / immunology
  • Autoimmunity
  • Biomarkers
  • Complement C3d / antagonists & inhibitors
  • Complement C3d / immunology*
  • Complement C3d / metabolism
  • Cytokines / metabolism
  • Disease Models, Animal
  • Epitopes, T-Lymphocyte / immunology
  • Female
  • Humans
  • Immunoglobulin G / immunology
  • Immunoglobulin G / metabolism
  • Inflammation Mediators
  • Ligands
  • Lupus Erythematosus, Systemic / drug therapy
  • Lupus Erythematosus, Systemic / immunology*
  • Lupus Erythematosus, Systemic / metabolism
  • Mice
  • Mice, Inbred MRL lpr
  • Mice, Knockout
  • Protein Binding / drug effects
  • Protein Binding / immunology

Substances

  • Antibodies, Monoclonal
  • Antigen-Antibody Complex
  • Autoantibodies
  • Biomarkers
  • Cytokines
  • Epitopes, T-Lymphocyte
  • Immunoglobulin G
  • Inflammation Mediators
  • Ligands
  • Complement C3d