Influence of the intravenous administration of ACTH-(1-24) on the characteristics of brain, heart and spleen adrenoceptors of haemorrhage-shocked rats

Pharmacol Res Commun. 1988 Sep;20(9):739-49. doi: 10.1016/s0031-6989(88)80714-8.

Abstract

Urethane-anesthetized rats were bled to otherwise irreversible haemorrhagic shock (mean arterial pressure = 18-25 mmHg) and then i.v. treated with ACTH-(1-24) (160 micrograms/kg) or saline. In comparison with sham-operated, non-shocked controls, bled rats showed a significant reduction in Bmax for [3H]Dihydroalprenolol and [3H]Dihydroergocryptine in heart ventricles, and for [3H]Yohimbine in spleen capsule. Neither the Kd of heart and spleen adrenoceptors nor the Bmax or Kd of brain adrenoceptors were affected. Treatment with ACTH-(1-24) restored to normal the Bmax for [3H]Dihydroalprenolol in heart ventricles, and for [3H]Yohimbine in the spleen capsule. These data indicate that the anti-shock effect of ACTH-(1-24) in bled rats is associated with a restoration of heart and spleen responsiveness to adrenergic stimuli.

MeSH terms

  • Animals
  • Brain / drug effects*
  • Cosyntropin / administration & dosage
  • Cosyntropin / pharmacology*
  • Dihydroalprenolol / metabolism
  • Heart / drug effects*
  • Injections, Intravenous
  • Kinetics
  • Myocardium / metabolism
  • Rats
  • Receptors, Adrenergic / metabolism*
  • Shock, Hemorrhagic / metabolism*
  • Spleen / drug effects*

Substances

  • Receptors, Adrenergic
  • Cosyntropin
  • Dihydroalprenolol