Activated PI3Kδ breaches multiple B cell tolerance checkpoints and causes autoantibody production

J Exp Med. 2020 Feb 3;217(2):e20191336. doi: 10.1084/jem.20191336.

Abstract

Antibody-mediated autoimmune diseases are a major health burden. However, our understanding of how self-reactive B cells escape self-tolerance checkpoints to secrete pathogenic autoantibodies remains incomplete. Here, we demonstrate that patients with monogenic immune dysregulation caused by gain-of-function mutations in PIK3CD, encoding the p110δ catalytic subunit of phosphoinositide 3-kinase (PI3K), have highly penetrant secretion of autoreactive IgM antibodies. In mice with the corresponding heterozygous Pik3cd activating mutation, self-reactive B cells exhibit a cell-autonomous subversion of their response to self-antigen: instead of becoming tolerized and repressed from secreting autoantibody, Pik3cd gain-of-function B cells are activated by self-antigen to form plasmablasts that secrete high titers of germline-encoded IgM autoantibody and hypermutating germinal center B cells. However, within the germinal center, peripheral tolerance was still enforced, and there was selection against B cells with high affinity for self-antigen. These data show that the strength of PI3K signaling is a key regulator of pregerminal center B cell self-tolerance and thus represents a druggable pathway to treat antibody-mediated autoimmunity.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, N.I.H., Intramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibody Formation / genetics*
  • Autoantibodies / blood
  • Autoantibodies / immunology*
  • Autoantigens / immunology
  • Autoimmunity / genetics
  • Class I Phosphatidylinositol 3-Kinases / blood
  • Class I Phosphatidylinositol 3-Kinases / genetics*
  • Class I Phosphatidylinositol 3-Kinases / metabolism
  • Female
  • Gain of Function Mutation*
  • Germinal Center / immunology
  • Humans
  • Immune Tolerance / immunology*
  • Immunoglobulin M / blood
  • Immunoglobulin M / immunology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Transgenic
  • Plasma Cells / immunology*
  • Signal Transduction / genetics

Substances

  • Autoantibodies
  • Autoantigens
  • Immunoglobulin M
  • Class I Phosphatidylinositol 3-Kinases
  • PIK3CD protein, human
  • Pik3cd protein, mouse