Netarsudil and latanoprost ophthalmic solution for the reduction of intraocular pressure in open-angle glaucoma or ocular hypertension

Expert Rev Clin Pharmacol. 2019 Dec;12(12):1073-1079. doi: 10.1080/17512433.2019.1701435.

Abstract

Introduction: Netarsudil and latanoprost ophthalmic solution (0.02%/0.005%) is indicated for intraocular pressure (IOP) lowering in open-angle glaucoma (OAG) or ocular hypertension (OHTN). The once-daily agent combines the mechanism of action for each of the individual components and provides a new avenue for long-term intraocular pressure control. This review aims to cover the agent's current efficacy and safety data and opine as to its role in glaucoma management.Areas covered: This article will cover Phase II-III clinical efficacy and safety data as well as basic science literature pertaining to the agent's mechanism of action and pharmacodynamics. In selecting articles for inclusion in this review, a literature search using the PubMed database was carried out. Cross-referencing was carried out where applicable. We did not use any date or language restrictions in electronic searches.Expert opinion: Netarsudil and latanoprost ophthalmic solution plays a pivotal role in management of individuals with OAG and OHTN. The agent may be used as first-line therapy to provide substantial IOP-lowering or when additional lowering is indicated and prostaglandins have provided insufficient IOP lowering. The once-daily dosing regimen decreases the risk of inadequate treatment due to nonadherence.

Keywords: Glaucoma treatment; latanoprost; netarsudil; rho-kinase inhibitor; trabecular meshwork.

Publication types

  • Review

MeSH terms

  • Animals
  • Antihypertensive Agents / administration & dosage
  • Antihypertensive Agents / adverse effects
  • Benzoates / administration & dosage*
  • Benzoates / adverse effects
  • Drug Combinations
  • Glaucoma, Open-Angle / drug therapy*
  • Humans
  • Intraocular Pressure
  • Latanoprost / administration & dosage*
  • Latanoprost / adverse effects
  • Ocular Hypertension / drug therapy*
  • Ophthalmic Solutions
  • beta-Alanine / administration & dosage
  • beta-Alanine / adverse effects
  • beta-Alanine / analogs & derivatives*

Substances

  • Antihypertensive Agents
  • Benzoates
  • Drug Combinations
  • Ophthalmic Solutions
  • beta-Alanine
  • Latanoprost
  • netarsudil