Phase II Study of Eribulin Mesylate Administered Biweekly in Patients With Human Epidermal Growth Factor Receptor-2-negative Metastatic Breast Cancer

Clin Breast Cancer. 2020 Apr;20(2):160-167. doi: 10.1016/j.clbc.2019.09.007. Epub 2019 Oct 14.

Abstract

Background: Patients with human epidermal growth factor receptor-2-negative metastatic breast cancer (MBC), whose disease progressed on prior chemotherapy, have a poor prognosis. Eribulin, a microtubule dynamics inhibitor, extends overall survival in previously treated MBC. The most common adverse event associated with eribulin is neutropenia, which may result in dose interruptions or reductions. A modified biweekly dosing schedule of eribulin was assessed for efficacy as well as improvements in hematologic toxicity.

Patients and methods: In this open-label, single-arm, multicenter, phase II study, previously treated (2-5 chemotherapy regimens for metastatic disease) patients with human epidermal growth factor receptor-2-negative MBC received intravenous eribulin 1.4 mg/m2 over 2 to 5 minutes on days 1 and 15 of each 28-day cycle. The primary study endpoints were objective response rate (ORR; complete response [CR] + partial responses [PR]) and disease control rate (DCR; CR + PR + stable disease [SD]).

Results: Among 58 treated patients, the ORR was 12% (95% confidence interval [CI], 5%-24%), DCR (CR, n = 1; PR, n = 6; SD, n = 30) was 65%, and the median progression-free survival was 3.6 months (95% CI, 2.9-4.1 months). Grade 3 or 4 neutropenia was 31%; 50% of all patients, and 78% of patients with neutropenia (all grades), received hematopoietic growth-factor support.

Conclusion: The efficacy and safety results obtained with a biweekly eribulin schedule in this phase II trial appear similar to those associated with the approved eribulin schedule (1.4 mg/m2 on days 1 and 8 of a 21-day cycle) reported in the EMBRACE study.

Keywords: Disease control rate; Dosing; HER2-negative; Objective response rate; Safety.

Publication types

  • Clinical Trial, Phase II
  • Multicenter Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Antineoplastic Agents / administration & dosage*
  • Antineoplastic Agents / adverse effects
  • Breast Neoplasms / drug therapy*
  • Breast Neoplasms / mortality
  • Breast Neoplasms / pathology
  • Drug Administration Schedule
  • Female
  • Furans / administration & dosage*
  • Furans / adverse effects
  • Granulocyte Colony-Stimulating Factor / administration & dosage
  • Humans
  • Injections, Intravenous
  • Ketones / administration & dosage*
  • Ketones / adverse effects
  • Middle Aged
  • Neutropenia / chemically induced
  • Neutropenia / diagnosis
  • Neutropenia / epidemiology*
  • Neutropenia / prevention & control
  • Prognosis
  • Progression-Free Survival
  • Receptor, ErbB-2 / analysis
  • Severity of Illness Index

Substances

  • Antineoplastic Agents
  • Furans
  • Ketones
  • Granulocyte Colony-Stimulating Factor
  • ERBB2 protein, human
  • Receptor, ErbB-2
  • eribulin