Oxidised metabolites of the omega-6 fatty acid linoleic acid activate dFOXO

Life Sci Alliance. 2020 Jan 28;3(2):e201900356. doi: 10.26508/lsa.201900356. Print 2020 Feb.

Abstract

Obesity-induced inflammation, or meta-inflammation, plays key roles in metabolic syndrome and is a significant risk factor in diabetes and cardiovascular disease. To investigate causal links between obesity, meta-inflammation, and insulin signaling we established a Drosophila model to determine how elevated dietary fat and changes in the levels and balance of saturated fatty acids (SFAs) and polyunsaturated fatty acids (PUFAs) influence inflammation. We observe negligible effect of saturated fatty acid on inflammation but marked enhancement or suppression by omega-6 and omega-3 PUFAs, respectively. Using combined lipidomic and genetic analysis, we show omega-6 PUFA enhances meta-inflammation by producing linoleic acid-derived lipid mediator 9-hydroxy-octadecadienoic acid (9-HODE). Transcriptome analysis reveals 9-HODE functions by regulating FOXO family transcription factors. We show 9-HODE activates JNK, triggering FOXO nuclear localisation and chromatin binding. FOXO TFs are important transducers of the insulin signaling pathway that are normally down-regulated by insulin. By activating FOXO, 9-HODE could antagonise insulin signaling providing a molecular conduit linking changes in dietary fatty acid balance, meta-inflammation, and insulin resistance.

MeSH terms

  • Animals
  • Animals, Genetically Modified
  • Cell Nucleus / metabolism
  • Chromatin / metabolism
  • Dietary Fats / adverse effects
  • Disease Models, Animal
  • Drosophila / genetics
  • Drosophila / metabolism*
  • Drosophila Proteins / genetics
  • Drosophila Proteins / metabolism*
  • Fatty Acids, Omega-3 / metabolism
  • Fatty Acids, Omega-3 / pharmacology
  • Forkhead Box Protein O3 / genetics
  • Forkhead Box Protein O3 / metabolism*
  • Forkhead Transcription Factors / genetics
  • Forkhead Transcription Factors / metabolism*
  • Gene Expression Regulation / drug effects
  • HeLa Cells
  • Humans
  • Inflammation / chemically induced
  • Inflammation / metabolism
  • Insulin / metabolism
  • Linoleic Acid / metabolism*
  • Linoleic Acid / pharmacology
  • Linoleic Acids, Conjugated / genetics
  • Linoleic Acids, Conjugated / metabolism
  • Linoleic Acids, Conjugated / pharmacology
  • Obesity / chemically induced
  • Obesity / metabolism*
  • Protein Binding
  • Signal Transduction / drug effects
  • Signal Transduction / genetics
  • Transcriptome
  • Transfection

Substances

  • Chromatin
  • Dietary Fats
  • Drosophila Proteins
  • FOXO protein, Drosophila
  • FOXO3 protein, human
  • Fatty Acids, Omega-3
  • Forkhead Box Protein O3
  • Forkhead Transcription Factors
  • Insulin
  • Linoleic Acids, Conjugated
  • 9-hydroxy-10,12-octadecadienoic acid
  • Linoleic Acid