DNA Nanostructures for Targeted Antimicrobial Delivery

Angew Chem Int Ed Engl. 2020 Jul 27;59(31):12698-12702. doi: 10.1002/anie.202002740. Epub 2020 May 20.

Abstract

We report the use of DNA origami nanostructures, functionalized with aptamers, as a vehicle for delivering the antibacterial enzyme lysozyme in a specific and efficient manner. We test the system against Gram-positive (Bacillus subtilis) and Gram-negative (Escherichia coli) targets. We use direct stochastic optical reconstruction microscopy (dSTORM) and atomic force microscopy (AFM) to characterize the DNA origami nanostructures and structured illumination microscopy (SIM) to assess the binding of the origami to the bacteria. We show that treatment with lysozyme-functionalized origami slows bacterial growth more effectively than treatment with free lysozyme. Our study introduces DNA origami as a tool in the fight against antibiotic resistance, and our results demonstrate the specificity and efficiency of the nanostructure as a drug delivery vehicle.

Keywords: DNA nanostructures; antimicrobial; atomic force microscopy; bionanotechnology; dSTORM.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Bacterial Agents / chemistry
  • Anti-Bacterial Agents / pharmacology*
  • Aptamers, Nucleotide / chemistry
  • Aptamers, Nucleotide / toxicity
  • Bacillus subtilis / chemistry
  • Bacillus subtilis / drug effects
  • COS Cells
  • Chlorocebus aethiops
  • DNA / chemistry*
  • DNA / toxicity
  • Drug Carriers / chemistry*
  • Drug Carriers / toxicity
  • Enzymes, Immobilized / chemistry
  • Enzymes, Immobilized / pharmacology
  • Escherichia coli / chemistry
  • Escherichia coli / drug effects
  • Microbial Sensitivity Tests
  • Muramidase / chemistry
  • Muramidase / pharmacology*
  • Nanostructures / chemistry*
  • Nanostructures / toxicity
  • Nucleic Acid Conformation

Substances

  • Anti-Bacterial Agents
  • Aptamers, Nucleotide
  • Drug Carriers
  • Enzymes, Immobilized
  • DNA
  • Muramidase