SIRT1-dependent mechanisms and effects of resveratrol for amelioration of muscle wasting in NASH mice

BMJ Open Gastroenterol. 2020 May;7(1):e000381. doi: 10.1136/bmjgast-2020-000381.

Abstract

Background: In non-alcoholic steatohepatitis (NASH), muscle wasting was an aggravating factor for the progression of hepatic steatosis. This study explores the potential benefits of chronic treatment with resveratrol, a strong activator of SIRT1 on the muscle wasting of NASH mice.

Methods: In vivo and in vitro study, we evaluate the SIRT1-dependent mechanisms and effects of resveratrol administration for 6 weeks with high-fat-methionine and choline deficient diet-induced NASH mice and palmitate-pretreated C2C12 myoblast cells.

Results: Resveratrol treatment improved grip strength and muscle mass of limbs, increased running distance and time on exercise wheels in NASH mice. There is a negative correlation between muscular SIRT1 activity and 3-nitrotyrosine levels of NASH and NASH-resv mice. The SIRT1-dependent effect of muscle wasting was associated with the suppression of oxidative stress, upregulation of antioxidants, inhibition of protein degradation, activation of autophagy, suppression of apoptotic activity, upregulation of lipolytic genes and the reduction of fatty infiltration in limb muscles of NASH mice. In vitro, resveratrol alleviated palmitate acid-induced oxidative stress, lipid deposition, autophagy dysfunction, apoptotic signals, and subsequently reduced fusion index and myotube formation of C2C12 cells. The beneficial effects of resveratrol were abolished by EX527.

Conclusions: Our study suggests that chronic resveratrol treatment is a potential strategy for amelioration of hepatic steatosis and muscle wasting in NASH mouse model.

Keywords: apoptosis; nonalcoholic steatohepatitis; oxidative stress; signalling.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antioxidants / metabolism
  • Apoptosis / drug effects
  • Autophagy / drug effects
  • Diet, High-Fat / adverse effects
  • Disease Models, Animal
  • Enzyme Inhibitors / administration & dosage
  • Enzyme Inhibitors / pharmacology
  • Enzyme Inhibitors / therapeutic use
  • Hand Strength / physiology
  • Mice
  • Mice, Inbred C57BL
  • Muscles / drug effects
  • Muscles / metabolism
  • Muscular Atrophy / drug therapy*
  • Muscular Atrophy / metabolism
  • Non-alcoholic Fatty Liver Disease / complications
  • Non-alcoholic Fatty Liver Disease / metabolism*
  • Oxidative Stress / drug effects
  • Resveratrol / administration & dosage
  • Resveratrol / pharmacology*
  • Resveratrol / therapeutic use
  • Sirtuin 1 / drug effects*
  • Sirtuin 1 / metabolism
  • Sirtuin 1 / pharmacology
  • Tyrosine / analogs & derivatives
  • Tyrosine / analysis
  • Up-Regulation

Substances

  • Antioxidants
  • Enzyme Inhibitors
  • 3-nitrotyrosine
  • Tyrosine
  • Sirt1 protein, mouse
  • Sirtuin 1
  • Resveratrol