Loss of the Ste20-like kinase induces a basal/stem-like phenotype in HER2-positive breast cancers

Oncogene. 2020 Jun;39(23):4592-4602. doi: 10.1038/s41388-020-1315-3. Epub 2020 May 11.

Abstract

HER2 is overexpressed in 20-30% of all breast cancers and is associated with an invasive disease and poor clinical outcome. The Ste20-like kinase (SLK) is activated downstream of HER2/Neu and is required for efficient epithelial-to-mesenchymal transition, cell cycle progression, and migration in the mammary epithelium. Here we show that loss of SLK in a murine model of HER2/Neu-positive breast cancers significantly accelerates tumor onset and decreases overall survival. Transcriptional profiling of SLK knockout HER2/Neu-derived tumor cells revealed a strong induction in the triple-negative breast cancer marker, Sox10, accompanied by an increase in mammary stem/progenitor activity. Similarly, we demonstrate that SLK and Sox10 expression are inversely correlated in patient samples, with the loss of SLK and acquisition of Sox10 marking the triple-negative subtype. Furthermore, pharmacological inhibition of AKT reduces SLK-null tumor growth in vivo and is rescued by ectopic Sox10 expression, suggesting that Sox10 is a critical regulator of tumor growth downstream of SLK/AKT. These findings highlight a role for SLK in negatively regulating HER2-induced mammary tumorigenesis and provide mechanistic insight into the regulation of Sox10 expression in breast cancer.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Transformation, Neoplastic / pathology*
  • Epithelial-Mesenchymal Transition / genetics
  • Female
  • Mice
  • Mice, SCID
  • Protein Serine-Threonine Kinases / genetics*
  • Protein Serine-Threonine Kinases / metabolism
  • Proto-Oncogene Proteins c-akt / antagonists & inhibitors
  • Receptor, ErbB-2 / metabolism*
  • SOXE Transcription Factors / genetics*
  • Spheroids, Cellular
  • Triple Negative Breast Neoplasms / genetics
  • Triple Negative Breast Neoplasms / pathology*
  • Tumor Cells, Cultured

Substances

  • SOXE Transcription Factors
  • Sox10 protein, mouse
  • Erbb2 protein, mouse
  • Receptor, ErbB-2
  • Protein Serine-Threonine Kinases
  • Proto-Oncogene Proteins c-akt
  • SLK protein, mouse

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