Steroid binding to cardiac type I receptors: in vivo studies

J Hypertens Suppl. 1988 Dec;6(4):S131-3. doi: 10.1097/00004872-198812040-00038.

Abstract

In vitro, Type I (mineralocorticoid) receptors show equivalently high affinity for aldosterone, corticosterone and cortisol in cytosol preparations from a wide range of tissues. This steroid non-selectivity is also found for hippocampal Type I receptors in vivo; in contrast, Type I receptors in physiological mineralcorticoid target tissues are highly aldosterone-specific in vivo. In the present study we show that Type I receptors in the heart are non-selective in vivo, like those in hippocampus, and therefore presumably act as high-affinity glucocorticoid receptors rather than mineralocorticoid receptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aldosterone / metabolism
  • Animals
  • Glucocorticoids / metabolism
  • Kidney / metabolism
  • Myocardium / metabolism*
  • Rats
  • Rats, Inbred Strains
  • Receptors, Steroid / classification
  • Receptors, Steroid / metabolism*

Substances

  • Glucocorticoids
  • Receptors, Steroid
  • Aldosterone