Evolution of Antimalarial Drug Resistance Markers in the Reservoir of Plasmodium falciparum Infections in the Upper East Region of Ghana

J Infect Dis. 2020 Oct 13;222(10):1692-1701. doi: 10.1093/infdis/jiaa286.

Abstract

Background: The majority of Plasmodium falciparum infections, constituting the reservoir in all ages, are asymptomatic in high-transmission settings in Africa. The role of this reservoir in the evolution and spread of drug resistance was explored.

Methods: Population genetic analyses of the key drug resistance-mediating polymorphisms were analyzed in a cross-sectional survey of asymptomatic P. falciparum infections across all ages in Bongo District, Ghana.

Results: Seven years after the policy change to artemisinin-based combination therapies in 2005, the pfcrt K76 and pfmdr1 N86 wild-type alleles have nearly reached fixation and have expanded via soft selective sweeps on multiple genetic backgrounds. By constructing the pfcrt-pfmdr1-pfdhfr-pfdhps multilocus haplotypes, we found that the alleles at these loci were in linkage equilibrium and that multidrug-resistant parasites have not expanded in this reservoir. For pfk13, 32 nonsynonymous mutations were identified; however, none were associated with artemisinin-based combination therapy resistance.

Conclusions: The prevalence and selection of alleles/haplotypes by antimalarials were similar to that observed among clinical cases in Ghana, indicating that they do not represent 2 subpopulations with respect to these markers. Thus, the P. falciparum reservoir in all ages can contribute to the maintenance and spread of antimalarial resistance.

Keywords: Plasmodium falciparum; Ghana; antimalarials; artemisinin-based combination therapies; asymptomatic reservoir; drug resistance; malaria; population genetics.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Aged, 80 and over
  • Alleles
  • Antimalarials / pharmacology*
  • Artemisinins / pharmacology
  • Child
  • Child, Preschool
  • Cross-Sectional Studies
  • Drug Resistance / drug effects*
  • Drug Resistance / genetics*
  • Female
  • Genetic Variation
  • Genetics, Population
  • Genotype
  • Ghana / epidemiology
  • Haplotypes
  • Humans
  • Infant
  • Malaria, Falciparum / epidemiology
  • Malaria, Falciparum / parasitology
  • Male
  • Membrane Transport Proteins
  • Middle Aged
  • Multidrug Resistance-Associated Proteins / genetics
  • Plasmodium falciparum / drug effects*
  • Plasmodium falciparum / genetics*
  • Protozoan Proteins / genetics
  • Young Adult

Substances

  • Antimalarials
  • Artemisinins
  • Mdr1 protein, Plasmodium falciparum
  • Membrane Transport Proteins
  • Multidrug Resistance-Associated Proteins
  • PfCRT protein, Plasmodium falciparum
  • Protozoan Proteins
  • artemisinin