Antagonistic effects of calcium ionophores and phorbol esters on T cell receptor mRNA levels in human thymocytes

J Immunol. 1988 Jan 15;140(2):361-6.

Abstract

Levels of mRNA of the T cell antigen receptors (TcR) in human thymocytes are differentially regulated in response to distinct intracellular signals. Activation of protein kinase C by the phorbol ester, tetradecanoyl phorbol acetate or other phorbol esters increases the levels of the alpha and beta T cell receptor (TcR-alpha, TcR-beta) mRNA, whereas an increase in cytosolic free Ca2+, induced by ionomycin or other Ca2+ ionophores, results in a decrease of alpha and beta TcR mRNA levels. In contrast, ionomycin increases the expression TcR-gamma mRNA whereas tetradecanoyl phorbol acetate prevents this induction. Our results suggest the existence of two opposing intracellular pathways that control expression of TcR-alpha and TcR-beta mRNA levels, on the one hand and TcR-gamma mRNA, on the other. These results provide the first evidence for antagonistic actions of protein kinase C and cytosolic-free Ca2+ on gene expression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Calcium / metabolism
  • Enzyme Activation / drug effects
  • Ethers / pharmacology
  • Gene Expression Regulation / drug effects
  • Humans
  • Ionomycin
  • Ionophores / pharmacology*
  • Nucleic Acid Hybridization
  • Protein Kinase C / metabolism
  • RNA, Messenger / antagonists & inhibitors*
  • Receptors, Antigen, T-Cell / analysis
  • Receptors, Antigen, T-Cell / drug effects*
  • Receptors, Antigen, T-Cell / genetics
  • T-Lymphocytes / drug effects
  • T-Lymphocytes / metabolism*
  • Tetradecanoylphorbol Acetate / pharmacology*

Substances

  • Ethers
  • Ionophores
  • RNA, Messenger
  • Receptors, Antigen, T-Cell
  • Ionomycin
  • Protein Kinase C
  • Tetradecanoylphorbol Acetate
  • Calcium