Production of colony-stimulating factor from macrophages by muroctasin

Arzneimittelforschung. 1988 Jul;38(7A):983-6.

Abstract

The effect of a muramyl dipeptide analog, N2-[(N-acetylmuramoyl)-L-alanyl-D-isoglutamyl]-N6-stearoyl-L-lysin e (MDP-Lys(L18), muroctasin), on the colony-stimulating factor (CSF) production was investigated in vitro. MDP-Lys(L18) stimulated murine peritoneal macrophages to induce CSF. However, the compound produced more CSF in the presence of both macrophages and T cell enriched fraction than in the absence of T cells. This phenomenon was found to be attributed to the fact that MDP-Lys(L18) also stimulated macrophages to induce interleukin 1 (IL-1) and the IL-1 induced CSF production by T cells. These findings suggest that macrophages may be the first target cells of MDP-Lys(L18) to produce CSF.

MeSH terms

  • Acetylmuramyl-Alanyl-Isoglutamine / analogs & derivatives*
  • Acetylmuramyl-Alanyl-Isoglutamine / pharmacology
  • Adjuvants, Immunologic / pharmacology*
  • Animals
  • Cell Line
  • Cells, Cultured
  • Colony-Stimulating Factors / biosynthesis*
  • Female
  • Interleukin-1 / biosynthesis
  • Macrophages / drug effects*
  • Macrophages / immunology
  • Macrophages / metabolism
  • Mice
  • T-Lymphocytes / immunology
  • T-Lymphocytes / metabolism

Substances

  • Adjuvants, Immunologic
  • Colony-Stimulating Factors
  • Interleukin-1
  • Acetylmuramyl-Alanyl-Isoglutamine
  • romurtide