HIV X4 Variants Increase Arachidonate 5-Lipoxygenase in the Pulmonary Microenvironment and are associated with Pulmonary Arterial Hypertension

Sci Rep. 2020 Jul 16;10(1):11696. doi: 10.1038/s41598-020-68060-9.

Abstract

Pulmonary Arterial Hypertension (PAH) is overrepresented in People Living with Human Immunodeficiency Virus (PLWH). HIV protein gp120 plays a key role in the pathogenesis of HIV-PAH. Genetic changes in HIV gp120 determine viral interactions with chemokine receptors; specifically, HIV-X4 viruses interact with CXCR4 while HIV-R5 interact with CCR5 co-receptors. Herein, we leveraged banked samples from patients enrolled in the NIH Lung HIV studies and used bioinformatic analyses to investigate whether signature sequences in HIV-gp120 that predict tropism also predict PAH. Further biological assays were conducted in pulmonary endothelial cells in vitro and in HIV-transgenic rats. We found that significantly more persons living with HIV-PAH harbor HIV-X4 variants. Multiple HIV models showed that recombinant gp120-X4 as well as infectious HIV-X4 remarkably increase arachidonate 5-lipoxygenase (ALOX5) expression. ALOX5 is essential for the production of leukotrienes; we confirmed that leukotriene levels are increased in bronchoalveolar lavage fluid of HIV-infected patients. This is the first report associating HIV-gp120 genotype to a pulmonary disease phenotype, as we uncovered X4 viruses as potential agents in the pathophysiology of HIV-PAH. Altogether, our results allude to the supplementation of antiretroviral therapy with ALOX5 antagonists to rescue patients with HIV-X4 variants from fatal PAH.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adult
  • Animals
  • Anti-HIV Agents / therapeutic use
  • Arachidonate 5-Lipoxygenase / metabolism*
  • Cells, Cultured
  • Cohort Studies
  • Disease Models, Animal
  • Endothelial Cells / metabolism
  • Female
  • Genotype
  • HIV Envelope Protein gp120 / genetics
  • HIV Infections / complications*
  • HIV Infections / drug therapy
  • HIV Infections / virology
  • HIV-1 / genetics*
  • HIV-1 / metabolism
  • Humans
  • Lung / metabolism*
  • Male
  • Middle Aged
  • Phenotype
  • Pulmonary Arterial Hypertension / complications*
  • Pulmonary Arterial Hypertension / virology
  • Pulmonary Artery / cytology
  • Rats
  • Rats, Inbred F344
  • Rats, Transgenic
  • Receptors, CXCR4 / metabolism
  • Viral Tropism / genetics*

Substances

  • Anti-HIV Agents
  • CXCR4 protein, human
  • HIV Envelope Protein gp120
  • Receptors, CXCR4
  • gp120 protein, Human immunodeficiency virus 1
  • Arachidonate 5-Lipoxygenase
  • ALOX5 protein, human