Exploring the Diversity of Cysteine-Rich Natural Product Peptides via MS/MS Fingerprint Ions

J Am Soc Mass Spectrom. 2020 Sep 2;31(9):1833-1843. doi: 10.1021/jasms.0c00078. Epub 2020 Jul 30.

Abstract

Natural product extracts present inherently complex matrices in which the identification of novel bioactive peptide species is challenged by low-abundance masses and significant structural and sequence diversity. Additionally, discovery efforts often result in the re-identification of known compounds, where modifications derived in vivo or during sample handling may obscure true sequence identity. Herein, we identify mass spectral (MS2) "fingerprint" ions characteristic of cyclotides, a diverse and biologically active family of botanical cysteine-rich peptides, based on regions of high sequence homology. We couple mass shift analysis with MS2 spectral fingerprint ions cross referenced with CyBase-a cyclotide database-to discern unique mass species in Viola communis extracts from mass species that are likely already characterized and those with common modifications. The approach is extended to a related class of cysteine-rich peptides, the trypsin inhibitors, using the characterized botanical species Lagenaria siceraria. Coupling the observation of highly abundant MS2 ions with mass shift analysis, we identify a new set of small, highly disulfide-bound cysteine-rich L. siceraria peptides.

MeSH terms

  • Cucurbitaceae / chemistry
  • Cyclotides* / analysis
  • Cyclotides* / chemistry
  • Cysteine / chemistry*
  • Disulfides / analysis
  • Plant Extracts* / analysis
  • Plant Extracts* / chemistry
  • Plant Proteins / analysis
  • Plant Proteins / chemistry
  • Tandem Mass Spectrometry / methods*
  • Trypsin Inhibitors / analysis
  • Trypsin Inhibitors / chemistry
  • Viola / chemistry

Substances

  • Cyclotides
  • Disulfides
  • Plant Extracts
  • Plant Proteins
  • Trypsin Inhibitors
  • Cysteine