Hydroxycocaines as Metabolic Indicators of Cocaine Ingestion

Forensic Sci Int. 2020 Dec:317:110516. doi: 10.1016/j.forsciint.2020.110516. Epub 2020 Sep 17.

Abstract

Hydroxycocaines in hair were investigated with many hundreds of head and body hair samples. All samples were washed by a published extensive aqueous method prior to confirmation by LC-MS/MS. Concentrations, percent of cocaine, and ratios of para- and meta-hydroxycocaines to ortho-hydroxycocaine are presented. Hydroxycocaines as percent of cocaine did not appear to be affected by cocaine concentrations, but were shown to increase with cocaethylene concentrations. Stability of hydroxycocaines over a year of ambient storage was demonstrated. Ortho-hydroxycocaine was shown to be formed by exposure of cocaine-positive hair to peroxide, while para- and meta-hydroxycocaines were not. Presence of para- or meta-hydroxycocaine at > 0.05% of cocaine is proposed as indicating ingestion of cocaine. This indicator prevents black hair from being more likely interpreted as positive for ingestion than lighter colored hair.

Keywords: Cocaethylene; Cocaine; Hair; Hydroxycocaines.

MeSH terms

  • Chromatography, Liquid
  • Cocaine / analogs & derivatives*
  • Cocaine / analysis*
  • Cocaine-Related Disorders / diagnosis*
  • Forensic Toxicology / methods
  • Hair / chemistry*
  • Humans
  • Limit of Detection
  • Mass Spectrometry
  • Specimen Handling
  • Substance Abuse Detection / methods*

Substances

  • Cocaine
  • 4'-hydroxycocaine