Synthesis of Indolizines from Pyridinium Salts and Ethyl Bromodifluoroacetate

Org Lett. 2020 Dec 4;22(23):9313-9318. doi: 10.1021/acs.orglett.0c03540. Epub 2020 Nov 16.

Abstract

Here we present a novel annulation of pyridinium salts with BrCF2CO2Et to access the indolizine derivatives with high efficiency. The α substitution of pyridine plays a key role in determining the reaction pathways. Various types of indolizines can be conveniently accessed from easily available pyridinium salts under mild and simple reaction conditions.

Publication types

  • Research Support, Non-U.S. Gov't