The deubiquitinase USP36 Regulates DNA replication stress and confers therapeutic resistance through PrimPol stabilization

Nucleic Acids Res. 2020 Dec 16;48(22):12711-12726. doi: 10.1093/nar/gkaa1090.

Abstract

PrimPol has been recently identified as a DNA damage tolerant polymerase that plays an important role in replication stress response. However, the regulatory mechanisms of PrimPol are not well defined. In this study, we identify that the deubiquitinase USP36 interferes with degradation of PrimPol to regulate the replication stress response. Mechanistically, USP36 is deubiquitinated following DNA replication stress, which in turn facilitates its upregulation and interaction with PrimPol. USP36 deubiquitinates K29-linked polyubiquitination of PrimPol and increases its protein stability. Depletion of USP36 results in replication stress-related defects and elevates cell sensitivity to DNA-damage agents, such as cisplatin and olaparib. Moreover, USP36 expression positively correlates with the level of PrimPol protein and poor prognosis in patient samples. These findings indicate that the regulation of PrimPol K29-linked ubiquitination by USP36 plays a critical role in DNA replication stress and chemotherapy response.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line, Tumor
  • Cisplatin / pharmacology
  • DNA Damage / drug effects
  • DNA Primase / genetics*
  • DNA Replication / drug effects*
  • DNA-Directed DNA Polymerase / genetics*
  • Deubiquitinating Enzymes / genetics
  • Drug Resistance, Neoplasm / drug effects
  • Drug Resistance, Neoplasm / genetics
  • Female
  • Gene Expression Regulation, Neoplastic / drug effects
  • Humans
  • Multifunctional Enzymes / genetics*
  • Ovarian Neoplasms / drug therapy
  • Ovarian Neoplasms / genetics*
  • Ovarian Neoplasms / pathology
  • Phthalazines / pharmacology
  • Piperazines / pharmacology
  • Polyubiquitin / genetics
  • Prognosis
  • Protein Stability / drug effects
  • Proteolysis / drug effects
  • Ubiquitin Thiolesterase / genetics*

Substances

  • Multifunctional Enzymes
  • Phthalazines
  • Piperazines
  • USP36 protein, human
  • Polyubiquitin
  • DNA Primase
  • PrimPol protein, human
  • DNA-Directed DNA Polymerase
  • Deubiquitinating Enzymes
  • Ubiquitin Thiolesterase
  • Cisplatin
  • olaparib