Histone H3.3G34-Mutant Interneuron Progenitors Co-opt PDGFRA for Gliomagenesis

Cell. 2020 Dec 10;183(6):1617-1633.e22. doi: 10.1016/j.cell.2020.11.012. Epub 2020 Nov 30.

Abstract

Histone H3.3 glycine 34 to arginine/valine (G34R/V) mutations drive deadly gliomas and show exquisite regional and temporal specificity, suggesting a developmental context permissive to their effects. Here we show that 50% of G34R/V tumors (n = 95) bear activating PDGFRA mutations that display strong selection pressure at recurrence. Although considered gliomas, G34R/V tumors actually arise in GSX2/DLX-expressing interneuron progenitors, where G34R/V mutations impair neuronal differentiation. The lineage of origin may facilitate PDGFRA co-option through a chromatin loop connecting PDGFRA to GSX2 regulatory elements, promoting PDGFRA overexpression and mutation. At the single-cell level, G34R/V tumors harbor dual neuronal/astroglial identity and lack oligodendroglial programs, actively repressed by GSX2/DLX-mediated cell fate specification. G34R/V may become dispensable for tumor maintenance, whereas mutant-PDGFRA is potently oncogenic. Collectively, our results open novel research avenues in deadly tumors. G34R/V gliomas are neuronal malignancies where interneuron progenitors are stalled in differentiation by G34R/V mutations and malignant gliogenesis is promoted by co-option of a potentially targetable pathway, PDGFRA signaling.

Keywords: GSX2; H3.3 G34R/V; PDGFRA; cell-of-origin; chromatin conformation; gliomas; interneuron progenitors; oncohistones; pediatric cancer; single-cell transcriptome.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Astrocytes / metabolism
  • Astrocytes / pathology
  • Brain Neoplasms / genetics*
  • Brain Neoplasms / pathology
  • Carcinogenesis / genetics*
  • Carcinogenesis / pathology
  • Cell Lineage
  • Cellular Reprogramming / genetics
  • Chromatin / metabolism
  • Embryo, Mammalian / metabolism
  • Epigenesis, Genetic
  • Gene Expression Regulation, Neoplastic
  • Gene Silencing
  • Glioma / genetics*
  • Glioma / pathology
  • Histones / genetics*
  • Histones / metabolism
  • Interneurons / metabolism*
  • Lysine / metabolism
  • Mice, Inbred C57BL
  • Models, Biological
  • Mutation / genetics*
  • Neoplasm Grading
  • Neural Stem Cells / metabolism*
  • Oligodendroglia / metabolism
  • Promoter Regions, Genetic / genetics
  • Prosencephalon / embryology
  • Receptor, Platelet-Derived Growth Factor alpha / genetics*
  • Receptor, Platelet-Derived Growth Factor alpha / metabolism
  • Transcription, Genetic
  • Transcriptome / genetics

Substances

  • Chromatin
  • Histones
  • Receptor, Platelet-Derived Growth Factor alpha
  • Lysine