[Antibacterial and antifungal compounds. VIII. Synthesis and antifungal activity of pyrrol derivatives similar to trichostatin A]

Farmaco Sci. 1987 Dec;42(12):893-903.
[Article in Italian]

Abstract

Some p-methylbenzolpyrrole acrylic acids and related compounds were synthesized. The new pyrrole derivatives have structural features in common with trichostatin A, an antifungal antibiotic. The above acids and derivatives were tested against Candida albicans and Candida sp in comparison with miconazole, pyrrolnitrin and amphotericin B and showed very weak antifungal activities. Occasionally some activity was found against a few strains of Candida albicans and against Candida pseudotropicalis.

MeSH terms

  • Antifungal Agents / chemical synthesis*
  • Antifungal Agents / pharmacology
  • Candida / drug effects
  • Candida albicans / drug effects
  • Chemical Phenomena
  • Chemistry
  • Hydroxamic Acids / chemical synthesis
  • Hydroxamic Acids / pharmacology
  • Microbial Sensitivity Tests
  • Pyrroles / chemical synthesis*
  • Pyrroles / pharmacology
  • Structure-Activity Relationship

Substances

  • Antifungal Agents
  • Hydroxamic Acids
  • Pyrroles
  • trichostatin A