MLH1 Deficiency-Triggered DNA Hyperexcision by Exonuclease 1 Activates the cGAS-STING Pathway

Cancer Cell. 2021 Jan 11;39(1):109-121.e5. doi: 10.1016/j.ccell.2020.11.004. Epub 2020 Dec 17.

Abstract

Tumors with defective mismatch repair (dMMR) are responsive to immunotherapy because of dMMR-induced neoantigens and activation of the cGAS-STING pathway. While neoantigens result from the hypermutable nature of dMMR, it is unknown how dMMR activates the cGAS-STING pathway. We show here that loss of the MutLα subunit MLH1, whose defect is responsible for ~50% of dMMR cancers, results in loss of MutLα-specific regulation of exonuclease 1 (Exo1) during DNA repair. This leads to unrestrained DNA excision by Exo1, which causes increased single-strand DNA formation, RPA exhaustion, DNA breaks, and aberrant DNA repair intermediates. Ultimately, this generates chromosomal abnormalities and the release of nuclear DNA into the cytoplasm, activating the cGAS-STING pathway. In this study, we discovered a hitherto unknown MMR mechanism that modulates genome stability and has implications for cancer therapy.

Keywords: DNA breaks; MLH1; RPA exhaustion; Rad51; cGAS-STING; chromosome instability; cytosolic DNA; exonuclease 1; mismatch repair.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line, Tumor
  • Chromosome Aberrations*
  • DNA Breaks, Single-Stranded
  • DNA Mismatch Repair
  • DNA Repair
  • DNA Repair Enzymes / metabolism*
  • DNA, Single-Stranded / metabolism
  • Exodeoxyribonucleases / metabolism*
  • HeLa Cells
  • Humans
  • Membrane Proteins / metabolism
  • Mice
  • MutL Protein Homolog 1 / deficiency*
  • MutL Protein Homolog 1 / metabolism
  • Neoplasms / genetics*
  • Neoplasms / metabolism
  • Nucleotidyltransferases / metabolism
  • Replication Protein A / metabolism
  • Signal Transduction*

Substances

  • DNA, Single-Stranded
  • MLH1 protein, human
  • Membrane Proteins
  • Replication Protein A
  • STING1 protein, human
  • Nucleotidyltransferases
  • cGAS protein, human
  • EXO1 protein, human
  • Exodeoxyribonucleases
  • MutL Protein Homolog 1
  • DNA Repair Enzymes