The Irradiated Brain Microenvironment Supports Glioma Stemness and Survival via Astrocyte-Derived Transglutaminase 2

Cancer Res. 2021 Apr 15;81(8):2101-2115. doi: 10.1158/0008-5472.CAN-20-1785. Epub 2021 Jan 22.

Abstract

The tumor microenvironment plays an essential role in supporting glioma stemness and radioresistance. Following radiotherapy, recurrent gliomas form in an irradiated microenvironment. Here we report that astrocytes, when pre-irradiated, increase stemness and survival of cocultured glioma cells. Tumor-naïve brains increased reactive astrocytes in response to radiation, and mice subjected to radiation prior to implantation of glioma cells developed more aggressive tumors. Extracellular matrix derived from irradiated astrocytes were found to be a major driver of this phenotype and astrocyte-derived transglutaminase 2 (TGM2) was identified as a promoter of glioma stemness and radioresistance. TGM2 levels increased after radiation in vivo and in recurrent human glioma, and TGM2 inhibitors abrogated glioma stemness and survival. These data suggest that irradiation of the brain results in the formation of a tumor-supportive microenvironment. Therapeutic targeting of radiation-induced, astrocyte-derived extracellular matrix proteins may enhance the efficacy of standard-of-care radiotherapy by reducing stemness in glioma. SIGNIFICANCE: These findings presented here indicate that radiotherapy can result in a tumor-supportive microenvironment, the targeting of which may be necessary to overcome tumor cell therapeutic resistance and recurrence. GRAPHICAL ABSTRACT: http://cancerres.aacrjournals.org/content/canres/81/8/2101/F1.large.jpg.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Astrocytes / enzymology*
  • Astrocytes / radiation effects
  • Brain / cytology
  • Brain / physiology
  • Brain / radiation effects*
  • Brain Neoplasms / pathology
  • Brain Neoplasms / radiotherapy*
  • Cell Survival / physiology
  • Enzyme Inhibitors / pharmacology
  • Extracellular Matrix / metabolism
  • Extracellular Matrix / radiation effects
  • Female
  • GTP-Binding Proteins / antagonists & inhibitors
  • GTP-Binding Proteins / metabolism*
  • Glioblastoma / pathology
  • Glioblastoma / radiotherapy*
  • Glioma / pathology
  • Glioma / radiotherapy
  • Humans
  • Male
  • Mice
  • Neoplasm Recurrence, Local / enzymology
  • Neoplasm Recurrence, Local / pathology
  • Neoplastic Stem Cells* / physiology
  • Protein Glutamine gamma Glutamyltransferase 2
  • Radiation Tolerance
  • Transglutaminases / antagonists & inhibitors
  • Transglutaminases / metabolism*
  • Tumor Microenvironment / physiology
  • Tumor Microenvironment / radiation effects*

Substances

  • Enzyme Inhibitors
  • TGM2 protein, human
  • Protein Glutamine gamma Glutamyltransferase 2
  • Transglutaminases
  • GTP-Binding Proteins