Angiogenesis in biliary tract cancer: targeting and therapeutic potential

Expert Opin Investig Drugs. 2021 Apr;30(4):411-418. doi: 10.1080/13543784.2021.1881479. Epub 2021 Mar 28.

Abstract

Introduction: Biliary Tract Cancer (BTC) is a heterogeneous group of malignant neoplasms with a complex molecular pathogenesis. The prognosis of metastatic disease is dramatically dismal and therapeutic options are scarce. Systemic chemotherapy is the gold standard for the metastatic disease. However, because of the disappointing results with conventional chemotherapy, investigators have turned to new biological therapeutic options targeting the main molecular pathways, neo-angiogenesis, involved in the disease pathogenesis.Areas covered: This paper examines the rationale of using antiangiogenic therapies in this setting, evaluates the therapeutic implications, and highlights ongoing studies and future perspectives. A Pubmed systematic review of preclinical and clinical data was performed which enabled the composition of this paper.Expert opinion: Amore in-depth understanding of the interplay between the neo-angiogenesis pathways, and the microenvironment will could propel the design new therapeutic strategies. Nowadays, the combination of antiangiogenic drugs and immune check-point inhibitors looks promising, but further, more comprehensive data are necessary to gain afuller picture. In an era of novel technologies and techniques, which includes radiomics, the challenge is to identify the biomarkers of response to antiangiogenic drugs which will permit the selection of patients that are more likely to respond to antiangiogenic therapies.

Keywords: Biliary tract cancer; anti-angiogenic drugs; bevacizumab; cholangiocarcinoma; immune checkpoint inhibitors; tyrosine-kinase inhibitors; vegf.

Publication types

  • Review

MeSH terms

  • Angiogenesis Inhibitors / administration & dosage
  • Angiogenesis Inhibitors / pharmacology*
  • Antineoplastic Combined Chemotherapy Protocols / administration & dosage
  • Antineoplastic Combined Chemotherapy Protocols / pharmacology
  • Biliary Tract Neoplasms / blood supply
  • Biliary Tract Neoplasms / drug therapy*
  • Humans
  • Immune Checkpoint Inhibitors / administration & dosage
  • Molecular Targeted Therapy
  • Neovascularization, Pathologic / drug therapy*
  • Neovascularization, Pathologic / pathology
  • Patient Selection
  • Prognosis
  • Tumor Microenvironment

Substances

  • Angiogenesis Inhibitors
  • Immune Checkpoint Inhibitors