[Phenotype- or genotype test for dihydropyrimidin dehydrogenase deficiency before treatment with a fluoropyrimidine]

Ugeskr Laeger. 2021 Feb 8;183(6):V07200556.
[Article in Danish]

Abstract

Some patients may have partial or complete deficiency of dihydropyrimidin dehydrogenase (DPD) and be more likely to experience severe toxicity with 5-fluorouracil. Since the spring of 2020, the Danish Medicines Agency has recommended genotype or phenotype testing before treatment with a fluoropyrimidine, but the most appropriate test strategy is debated. In this review, we present polymorphisms in the genes coding for DPD and summarise the evidence for DPD-enzyme deficiency testing and pharmacokinetic guided dosing.

Publication types

  • Review

MeSH terms

  • Antimetabolites, Antineoplastic / therapeutic use
  • Dihydropyrimidine Dehydrogenase Deficiency* / drug therapy
  • Dihydropyrimidine Dehydrogenase Deficiency* / genetics
  • Dihydrouracil Dehydrogenase (NADP) / genetics
  • Fluorouracil / adverse effects
  • Genotype
  • Humans
  • Phenotype

Substances

  • Antimetabolites, Antineoplastic
  • Dihydrouracil Dehydrogenase (NADP)
  • Fluorouracil